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5-[(3R,4R)-4-(azepan-1-yl)-3-hydroxypiperidine-1-carbonyl]-1,2-dihydropyridin-2-one
9-[(4,5-dichlorothiophen-2-yl)sulfonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
2-(2-phenylethyl)-8-(pyridazine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
dimethyl({2-[1-(thiophene-3-sulfonyl)piperidin-2-yl]ethyl})amine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
4-benzyl-1-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}piperidine
1-(cyclohexylmethyl)-N-ethyl-5-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]imidazo[1,2-a]pyrimidine-2-carboxamide
1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
(3aR,7aS)-5-methyl-2-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
9-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane
5-({[2-(dimethylamino)-6-ethylpyrimidin-4-yl]amino}methyl)-N,N-dimethylfuran-2-carboxamide
(3S,4R)-1-[3-(azocan-1-yl)propanoyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
3-(4-methyl-1,3-thiazol-5-yl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]propanamide
1-[(2-ethoxypyridin-3-yl)methyl]-3-(2,4,6-trimethylpyridin-3-yl)urea
(butan-2-yl)[(4-methanesulfonylphenyl)methyl](thiophen-3-ylmethyl)amine
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2-{[2-amino-6-(2-methoxyquinolin-3-yl)pyrimidin-4-yl]amino}ethan-1-ol
6-[(diethylamino)methyl]-N-[(3-methylpyridin-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-2,3-dihydro-1H-isoindole
methyl (1R,3S,3aR,6aS)-3-(5-chlorothiophen-2-yl)-1-ethyl-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N3-(adamantan-1-ylmethyl)-N5-[1-(furan-2-yl)ethyl]-N3-methyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(4-methylphenyl)-4-[2-(2-oxopyrrolidin-1-yl)propanoyl]piperazin-2-one
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]naphthalene-1-carboxamide
4-(4-chlorophenyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]butanamide
N-[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]-2-(1H-imidazol-2-yl)benzamide
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
2-amino-N-[1-(4-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]acetamide
1-(but-3-en-1-yl)-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
1-(propan-2-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine-4-carboxamide
1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(4H-1,2,4-triazol-4-yl)propan-1-one
N-[(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
3-(1-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)-1,2-dihydroquinolin-2-one
8-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
N-(2-methyl-1,3-benzothiazol-5-yl)-6-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(benzylsulfanyl)ethyl]-1-(pyridin-2-yl)piperidine-3-carboxamide
9-(3-fluoro-4-methylbenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-[4-(propan-2-yl)phenyl]urea
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
N-[(2R,3R)-1'-[(2,3-dimethoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
1-(2-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
3-[(3-cyanopiperidin-1-yl)sulfonyl]-N-(1,2-oxazol-3-ylmethyl)benzamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
{2-[3-(trifluoromethyl)phenyl]-1,3-thiazol-4-yl}methanol
(1R,2S)-1-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-2,3-dihydro-1H-inden-2-ol
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-methoxypyrimidine
N-(isoquinolin-5-ylmethyl)-N,2,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-(4-chlorophenoxy)-1-[3-(methylsulfanyl)propyl]piperidine-4-carboxylic acid
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide