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1-[1-(2,2-dimethylpropyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]-2-(3-fluorophenyl)piperidine
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](ethyl)(oxan-4-ylmethyl)amine
1-(1,1-dioxo-1λ6-thiane-4-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
5-(dimethylamino)-2-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-2,3-dihydropyridazin-3-one
3-{1-[2-(2-oxopiperidin-1-yl)acetyl]piperidin-4-yl}-N-phenylpropanamide
(2S,4S)-4-amino-1-[2-(1H-imidazol-2-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(1,4-dioxan-2-ylmethyl)-N-methyl-5-(naphthalen-2-yl)-1,2,4-triazin-3-amine
methyl 5-(cycloheptylamino)-3-acetamido-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-6-(trifluoromethyl)pyridine-3-carboxamide
4-[3-(3-chlorophenyl)pyrrolidine-1-carbonyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-[(naphthalen-1-ylmethyl)amino]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N,2-dimethyl-N-[(4-phenylphenyl)methyl]-1,3-thiazole-4-carboxamide
1-({1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-3-yl}methyl)pyrrolidin-2-one
3-{5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
8-(2-butoxybenzoyl)-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(5-methylthiophen-2-yl)methyl]piperidine
N-(pyrrolidin-3-yl)-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
2-({2-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-methoxypropyl)acetamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[4-(1H-pyrazol-3-yl)benzoyl]-1,4-diazepane
5-[3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoxaline
1-(1H-imidazol-4-ylmethyl)-4-(2-phenoxyethyl)piperazine
4-cyclobutanecarbonyl-N-[2-(2-methylpropoxy)phenyl]-1,4-diazepane-1-carboxamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
1,7-dimethyl-5-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-2,4-dione
5-(1-ethyl-1H-imidazol-2-yl)-1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-phenyl-1H-imidazole
N-[(3-methoxyphenyl)methyl]-6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-methyl-N-({5-[(2-phenylmorpholin-4-yl)methyl]furan-2-yl}methyl)methanesulfonamide
4-ethyl-3-[1-(pyrrolidine-1-sulfonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(7-methyl-1-benzofuran-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-cyclopentanecarbonyl-4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}piperidine
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-[(2-chlorophenyl)methyl]-N-(oxan-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)pent-4-enamide
N-phenyl-2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
(2S)-2-{[2-(dimethylamino)-4-methylpyrimidin-5-yl]formamido}-3-(4-hydroxyphenyl)propanamide
N-[2-(1H-imidazol-4-yl)ethyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
5-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyrazin-2-amine
4-[5-(ethoxymethyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
2-(2-chloro-4-fluorophenoxymethyl)-4-(3-propylpyrrolidine-1-carbonyl)-1,3-oxazole
4-{5-[2-(1H-imidazol-2-yl)phenyl]-3-methyl-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
4-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
10-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carbonitrile
3-(pyrrolidin-1-ylmethyl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-ol
2-methyl-8-(1H-1,2,4-triazole-5-carbonyl)-2,8-diazaspiro[4.5]decane
N-[2-(1,3-benzothiazol-2-yl)ethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
ethyl 4-[(2-chlorophenyl)methyl]-1-[2-(4-ethylpiperazin-1-yl)acetyl]piperidine-4-carboxylate