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1-acetyl-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylpiperidine-4-carboxamide
N-methyl-5-{1-[3-(methylsulfanyl)propyl]pyrrolidin-2-yl}-N-(pyrazin-2-ylmethyl)thiophene-2-carboxamide
N-(1,4-dioxan-2-ylmethyl)-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanamide
1-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-4-(3-methylpyridin-4-yl)piperazine
N-[2-(4-methoxyphenyl)ethyl]-N-(oxolan-2-ylmethyl)-2-(2-oxopiperidin-1-yl)acetamide
6-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(2-fluorophenoxy)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine-4-carboxylic acid
4-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1λ6-thiomorpholine-1,1-dione
N-cyclopropyl-3,4-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-5-sulfamoylbenzamide
(1S,5R)-3-{2-[4-(dimethylamino)phenyl]acetyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2-[(4-chlorophenyl)methoxy]ethyl}-4-methylpiperidine-4-carboxamide
1-[2-(dimethylamino)ethyl]-3-(3-methoxyphenyl)-3-{2-oxo-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
N-(1-methoxypropan-2-yl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
6,7-dimethyl-4-({[2-(pyridin-2-yl)ethyl]amino}methyl)-2H-chromen-2-one
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]pyrimidin-2-amine
1-ethyl-4-{[3-(3-ethylphenoxy)azetidin-1-yl]methyl}-1H-pyrazole
4-(3-hydroxy-3-methylbutyl)-N-[1-(4-hydroxyphenyl)ethyl]benzamide
methyl 2-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methylacetamido]acetate
4-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-3-yl]-2-methyl-6-(pyrrolidin-1-yl)pyrimidine
N-{[1-(7-fluoro-2-methylquinoline-4-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
1-(2-aminoethyl)-N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-({3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}methyl)-2-methoxyphenoxy]acetamide
3-hexyl-8-[(2R)-pyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,4-dimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
3-(pyridin-2-yl)-N-[(2R)-pyrrolidin-2-ylmethyl]-1H-pyrazole-5-carboxamide
4-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-N-(propan-2-yl)pyridine-2-carboxamide
1-(3-fluorobenzoyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(thiophen-2-yl)acetamide
2-ethyl-4-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}pyrimidine
N-(2,2-dimethyloxan-4-yl)-N-ethyl-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetamide
(4aS,7aR)-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{3-[(3-chlorophenyl)methyl]-1-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
6-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-4-amine
2-{4-[(4-fluoro-3-methoxyphenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
1-[(3S)-3-(dimethylamino)azepan-1-yl]-3-{[(4-fluorophenyl)methyl]sulfanyl}propan-1-one
N3-(butan-2-yl)-1-cyclopentyl-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(1R,3S)-3-methoxy-7-(3-methoxybenzenesulfonyl)-7-azaspiro[3.5]nonan-1-ol
6-methyl-2-phenyl-N-[2-(pyridin-4-yl)ethyl]pyrimidin-4-amine
2-{[(1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)oxy]methyl}pyridine
3-{2-[3-(cyclopentylcarbamoyl)propanamido]ethoxy}benzoic acid
6,8-dimethyl-2-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-1,4-dihydroquinolin-4-one
1-[(1S,5R)-6-(8-chloro-2-methylquinoline-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-cyclopentyl-2-{methyl[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]amino}propanamide
1-ethyl-N-[2-(2-fluorophenyl)ethyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(1-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
(3S,4R)-1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[1-(4-fluorophenyl)propyl]propanamide
dimethyl({[4-methyl-5-(1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
(3S,4S)-1-(5-ethyl-1,2-oxazole-3-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
4-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}-3-methylpiperazin-2-one