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2-[4-(ethylsulfanyl)phenyl]-2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]acetic acid
2-({4-[5-(aminomethyl)thiophen-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
(1R,3S)-7-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-7-azaspiro[3.5]nonane-1,3-diol
6-(2,5-dimethylphenyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(4-methoxyphenyl)-5-{1H-pyrrolo[2,3-b]pyridin-1-ylmethyl}-1,2,4-oxadiazole
N-[(2R,3R)-1'-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-(2-chlorophenyl)-N,3-dimethyl-N-(2-methylpropyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[4-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperazin-1-yl]ethan-1-ol
4-(2-methyl-1,3-thiazole-4-carbonyl)-7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-propyl-4-[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]aniline
2-[4-(3-cyclopentylpropyl)-1-methylpiperazin-2-yl]ethan-1-ol
4,6-dimethyl-1-(2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
2-[1-(2-methylpropyl)-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl]ethan-1-ol
N-methyl-5-[(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]furan-2-carboxamide
N-(4-{3-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidine-1-carbonyl}phenyl)acetamide
4-methyl-3-{[(oxolan-3-yl)carbamoyl]amino}-N-propylbenzamide
1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-methyl-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
2-(2,3-dimethylphenoxy)-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]ethan-1-one
1-{spiro[2.3]hexane-1-carbonyl}-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
1-(2-methoxyethyl)-N-[(1-methylpiperidin-4-yl)methyl]-5-oxo-N-(2-phenylethyl)pyrrolidine-3-carboxamide
3-[2-(4-methylpiperazin-1-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-6-methyl-2-propylpyrimidine
2-(4-fluorophenyl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidine
1-[(2-methylphenyl)methyl]-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
(2S,4R)-4-amino-N,N-diethyl-1-{2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidine-2-carboxamide
(1S,5R)-3-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[1-(5-ethyl-1,3,4-thiadiazol-2-yl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
methyl 6-[(thiomorpholine-4-carbonyl)amino]-1,2,3,4-tetrahydroquinoline-1-carboxylate
methyl 5-(2-methanesulfonamidopropanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[(4-fluorophenyl)methyl]-3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)propanamide
2-[({1-[(2-chloro-6-fluorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}methyl)sulfanyl]pyrimidine
3-chloro-N-cyclopentyl-4-({1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}oxy)benzamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-(2,5-dioxoimidazolidin-4-yl)-N-methylpropanamide
[(3R,4S)-1-(2,2-diphenylethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
[2-(4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}phenoxy)ethyl]dimethylamine
3-({1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
4-fluoro-N-[2-(7-{[2-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
5-({5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}methyl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
4-[4-({methyl[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)phenyl]but-3-yn-1-ol
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-[3-(1H-1,2,3-triazol-1-yl)propyl]propanamide
(3S,4S)-4-(4-benzylpiperazin-1-yl)-1-(2-methylfuran-3-carbonyl)pyrrolidin-3-ol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(2-oxo-1,3-oxazolidin-5-yl)methyl]piperidine-4-carboxamide
6-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
(3S,7S)-5-[2-(dimethylamino)benzoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
6-fluoro-2-{[3-(propoxymethyl)pyrrolidin-1-yl]methyl}quinolin-4-ol
(3S)-1-ethyl-3-methyl-4-(3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperazin-2-one
(benzylsulfamoyl)({[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amine
N,N-dimethyl-7-(4-methylbenzoyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine