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N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3-(1H-pyrazol-4-yl)benzamide
3-(2-fluorophenoxymethyl)-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
2-{3-[4-(3-methylpyridin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}acetamide
1-ethyl-4-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine
N-[(7-{[4-(dimethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-2-(3-fluorophenyl)acetamide
1-(cyclohexylmethyl)-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
1-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
1-cyclobutanecarbonyl-4-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)piperidine
1-(2,3-dimethoxyphenyl)-2-(3-methylfuran-2-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-ethyl-N-[2-(morpholin-4-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
4-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]-2,6-dimethylpyrimidine
2-cyclopentyl-N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
(3S)-1-(5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)pyrrolidin-3-ol
4-{5-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)methyl]thiophen-2-yl}-2-methylbut-3-yn-2-ol
2-methyl-4-{4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
4-(4-chlorophenoxy)-1-(pyridin-2-ylmethyl)piperidine-4-carboxylic acid
1-{[2-chloro-5-methoxy-4-(propan-2-yloxy)phenyl]methyl}pyrrolidin-3-amine
1-(2-{[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]amino}ethyl)imidazolidin-2-one
6-{2-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-2-methylpyrimidin-4-ol
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-4-ethyl-1,3-thiazol-2-amine
1-{2-[4-(3-propoxypiperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}piperazine
N-cyclopentyl-1-methyl-N-[(5-methylthiophen-2-yl)methyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-[(2-chloro-4-fluorophenyl)methyl]-N-[2-(cyclohex-1-en-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-ethyl-2,5-dimethyl-1H-pyrrole-3-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}propanamide
N-[(2,5-dimethylphenyl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
9-(3-propyl-1H-pyrazole-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(cyclobutylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(1H-imidazol-1-yl)propan-1-one
2-(3-fluorophenoxymethyl)-N-[(2-methylphenyl)methyl]-1,3-oxazole-4-carboxamide
1-[(2-chloro-6-fluorophenyl)methyl]-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazole
methyl 3-cyclobutaneamido-5-{[(4-methoxy-3-methylphenyl)methyl]amino}-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]pyrazin-2-ol
2-[(5-methylpyrazin-2-yl)methyl]-9-(4-methylpyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(methoxymethyl)-N-[(3R,4S)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]cyclobutane-1-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-hexyl-8-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[(8-methoxyquinolin-2-yl)methyl](methyl)[2-(pyridin-4-yl)ethyl]amine
4-({[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}(methyl)amino)-1λ6-thiane-1,1-dione
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(2E)-N-cyclopropyl-3-(3,4-dimethoxyphenyl)-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)prop-2-enamide
N-[5-(2-methoxyacetamido)-2-methylphenyl]-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
11-(5-chloropyridine-2-carbonyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(1,3-dihydroxy-2-methylpropan-2-yl)acetamide
N,4-dimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3-thiadiazole-5-carboxamide
4-{[(2-methoxyphenyl)methyl]amino}-5-methyl-N-(quinolin-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide