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N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-2-(piperidin-1-yl)acetamide
4-(2,6-dimethylpyridin-3-yl)-2-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidine
N-{2-[(2,5,7-trimethylquinolin-4-yl)formamido]ethyl}acetamide
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]-1,3-benzothiazole
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
1-[(3-fluorophenyl)methyl]-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
N-cyclopropyl-15-methyl-13-oxo-9-(pyridin-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
1-(2-benzylmorpholin-4-yl)-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
4-{1-[3-(1-methylcyclopropyl)propanoyl]piperidin-3-yl}benzoic acid
3-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(2-methyl-2H-1,2,3-benzotriazol-4-yl)urea
3-methyl-1-{1-[6-(quinolin-8-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
1-(4-benzylpiperidin-1-yl)-3-[1-(thiophene-2-carbonyl)piperidin-4-yl]propan-1-one
1-methyl-4-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)-1,4-diazepane
1-[(3-chlorophenyl)methyl]-4-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
1-[(3-{2-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]ethoxy}-4-methoxyphenyl)methyl]-4-(4-fluorophenyl)piperazine
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-(2-methyl-2,3-dihydro-1H-indol-1-yl)ethane-1,2-dione
N-[5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]-4-(morpholine-4-carbonyl)piperazine-1-carboxamide
(4aS,8aR)-6-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[5-(3-fluorophenyl)-1H-indazol-1-yl]acetamide
N-benzyl-N-(1,3-thiazol-2-ylmethyl)morpholine-2-carboxamide
methyl 4-oxo-4-(4-{3-[(pyridin-2-ylmethyl)carbamoyl]phenoxy}piperidin-1-yl)butanoate
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-sulfamoylbenzamide
2-[1-(2-methylpropyl)-4-[(2,4,5-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
5-(4-methoxy-2-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-{1-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
2-ethyl-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)butanamide
methyl (2S,4R)-1-[(4-ethoxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
N-[(1R,3S)-3-{[(3-fluorophenyl)methyl]carbamoyl}cyclopentyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
8-[2-(2-oxopyrrolidin-1-yl)ethyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-methoxy-N,3-dimethyl-1-benzofuran-2-carboxamide
3-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-(2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
5-[1-(2,3-dihydro-1H-inden-2-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})amine
2-(3-hydroxyphenyl)-N-{[1-(pyridin-3-ylmethyl)piperidin-4-yl]methyl}acetamide
2-[2-(dimethylamino)ethyl]-8-[3-(2-fluorophenyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
6-{4-[1-(morpholin-4-yl)ethyl]phenyl}-2-(pyrrolidin-1-yl)pyrimidin-4-amine
1'-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]spiro[indene-1,4'-piperidine]
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-(thiophen-2-yl)butanamide
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-{thieno[3,2-d]pyrimidin-4-yl}-decahydroisoquinoline
4-(4-chlorophenyl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}butanamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-[(1s,5s)-7,10-dimethyl-3,7,10-triazatricyclo[3.3.3.01,5]undecan-3-yl]ethan-1-one
methyl 3-(2,4-dimethoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxylate
3-{imidazo[1,2-a]pyridin-2-yl}-5-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazole
8-{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one