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(1R,6S)-N-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
7-(phenoxathiin-4-yl)-4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrol-2-yl]-6-methylpyrimidin-2-yl}phenol
(4-{[1-(thiophen-3-yl)ethyl]amino}quinazolin-2-yl)methanol
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-(oxolan-3-yl)benzamide
methyl 3-[(2E)-3-(2-fluorophenyl)prop-2-enamido]-6-{[methyl(propan-2-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-({7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(2-phenoxyethyl)piperazine
4-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-({1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1,3-thiazole
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
2-(1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)benzoic acid
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(4-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
1-(1-{[3-(morpholin-4-ylmethyl)phenyl]methyl}piperidin-4-yl)piperidin-3-ol
(2E)-N-{[7-(dimethyl-1,3-thiazole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
1-(4-ethylpiperazin-1-yl)-3-[3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
[(4-fluorophenyl)methyl](methyl){[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
2-{1-[2-(3-methoxyphenyl)ethyl]-1H-imidazol-2-yl}-4-methyl-1,3-thiazole
2-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-4-(trifluoromethyl)pyridine
4,6-dimethyl-N-[2-(2-methylpropanesulfonyl)ethyl]pyrimidin-2-amine
N-[(3R,4R)-3-hydroxy-1-{[5-(4-methylphenyl)furan-2-yl]methyl}piperidin-4-yl]pyridine-3-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]propanamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[1-(4-methoxyphenyl)ethyl]-N-methyl-1,2-oxazole-3-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(2-methylfuran-3-carbonyl)pyrrolidin-3-yl]methanol
5-{cyclopropyl[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1-methyl-1H-1,2,4-triazole
1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
4-[(4-methylphenyl)methyl]-3-{2-oxo-2-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethyl}piperazin-2-one
6-acetamido-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)pyridine-3-carboxamide
N-(2-hydroxyethyl)-1-methyl-N-[(2-methylphenyl)methyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
4-({2-[(benzenesulfonyl)methyl]phenyl}methyl)-1,3λ6,4-oxathiazinane-3,3-dione
2-[1-(2,2-dimethylpropyl)-4-{[2-(furan-2-yl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
1-(3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzoyl)azepane
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
(1s,4s)-4-{8-benzyl-2,8-diazaspiro[5.5]undecane-2-carbonyl}cyclohexan-1-ol
5-(5-chloro-2-methoxyphenyl)-3-cyclobutyl-1H-1,2,4-triazole
1-(1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
3-(3-methoxyphenoxymethyl)-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperidine
8-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
(3S,4R)-1-methanesulfonyl-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
(2S)-N-(3-carbamoyl-4-fluorophenyl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
N-[1-(2-methoxyphenyl)propan-2-yl]-N-methylquinoxaline-5-carboxamide
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methylpiperidine
8-[(5-ethylpyridin-2-yl)methyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
{1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-4-yl}(thiophen-2-yl)methanol
1-(3-methylpyridin-2-yl)-4-[3-(methylsulfanyl)butyl]piperazine
9-methoxy-3-[(4-methoxy-2,3-dimethylphenyl)methyl]-N-methyl-7-oxo-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidine-3-carboxamide
5-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}isoquinoline