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[1-(4-methanesulfonylbenzoyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
1,3,5-trimethyl-4-[1-methyl-5-(2-phenylpyrrolidine-1-carbonyl)-1H-pyrazol-3-yl]-1H-pyrazole
2-[(2,1,3-benzoxadiazol-5-ylmethyl)amino]-N-phenylbutanamide
methyl (2S)-2-{[5-(cyclooctylcarbamoyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridin-3-yl]formamido}-3-methylbutanoate
3-(1-ethyl-1H-imidazol-2-yl)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
2-(2-{[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-{1-[(1-benzofuran-5-yl)carbamoyl]pyrrolidin-3-yl}benzoic acid
3,5-dimethyl-1-({3-[2-(2-phenylethyl)pyrrolidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-pyrazole
3-(4-{[3-(1H-1,3-benzodiazol-2-yl)azetidin-1-yl]methyl}phenyl)prop-2-yn-1-ol
1-(1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)propan-1-one
(3R,4R)-4-amino-1-{5-[(diethylamino)methyl]-2-phenylfuran-3-carbonyl}piperidin-3-ol
N-[(2R,3R)-1'-[(2-chloro-6-fluorophenyl)methyl]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
(3R,4R)-4-ethyl-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidine-3,4-diol
(5S,9aS,9bS)-5-(isoquinolin-5-yl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propanoyl)-6-[(4-fluorophenyl)methoxy]-1-(propan-2-yl)-1,4-diazepan-2-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-(4-carbamoyl-3-chlorophenyl)-N,N-dimethylpyridine-3-carboxamide
ethyl 1-{[3-(2-hydroxyethoxy)phenyl]methyl}-3-(2-phenoxyethyl)piperidine-3-carboxylate
2-amino-6-methyl-4-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-methoxy-N-[2-(1,3-oxazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
propan-2-yl 2-[(3-methoxyphenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxylate
(4aS,7aR)-1-(1-ethylpiperidine-4-carbonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2-chloro-4-fluorophenyl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-1-cyclopentylpiperidin-2-one
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
1-benzyl-N-ethyl-5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
5-ethyl-4-(3-phenylpiperazin-1-yl)pyrimidin-2-amine
1-(2-methoxy-5-{[(pyridin-4-ylmethyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
3-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine-4-carbonyl}-N-methylpyridin-2-amine
1-(4-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-one
2,5-dimethyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-ethyl-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(5-methylfuran-2-yl)methyl]piperidine
3-(2-methoxyphenyl)-1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]propan-1-one
1-(3-phenylpropyl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}piperidin-2-one
1,6-dimethyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-3-(4-methoxyphenyl)propan-1-ol
methyl 1-[(3R,5S)-1-[(4-methoxyphenyl)methyl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-{4-methoxy-3-[2-(morpholin-4-yl)ethoxy]phenyl}-1H-1,3-benzodiazole
2-(2-{1-[4-(1H-pyrazol-4-yl)butanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
3-[({5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}amino)methyl]-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
5-cyclobutanecarbonyl-1'-(3-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(2-benzyl-1,3-thiazole-4-carbonyl)-2-phenylmorpholine
9-[2-(propan-2-yloxy)propanoyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-1H,3H,4H,5H-thiopyrano[4,3-b]indole-8-carboxamide
3-{[1-(3-methylbut-2-enoyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
1-(cyclopropylmethyl)-3-(2-methylquinolin-5-yl)-6-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-cyclopentyl-2-{[(3,4-dichlorophenyl)methyl]amino}propanamide