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4-({ethyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-N-(1,2,3-thiadiazol-5-yl)benzamide
N-[2-(2-chloro-6-methylphenoxy)ethyl]-2,2-dimethyloxane-4-carboxamide
(2S,4S)-1-(cyclohexylmethyl)-N-[2-(2-methoxyphenyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N3-butyl-1-cyclohexyl-N5-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-methoxyethyl)-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
3-{imidazo[1,2-a]pyridin-3-ylmethyl}-3H,4H-pyrido[3,4-d]pyrimidin-4-one
N-[1-ethyl-2-(3-methoxyphenyl)-7-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl]acetamide
N-[(1-propyl-1H-imidazol-2-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-[3-chloro-2-(4-ethylpiperazin-1-yl)phenyl]oxolane-2-carboxamide
(1S,5R)-6-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
(1R,5R)-3-(2-chloro-4-fluorobenzenesulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-4-(thian-4-yl)piperazine
1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1,4-diazepane-6-carboxylic acid
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
1-(2-{[(2,2-dimethylpropyl)(methyl)amino]methyl}-6-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
(2S)-2-({4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}amino)butan-1-ol
6-{[2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]sulfonyl}-2,3-dihydro-1,3-benzothiazol-2-one
3-(1-ethyl-1H-imidazol-2-yl)-1-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidine
2-[(3S,4R)-3-propyl-4-[2-(pyrrolidin-1-yl)benzamido]pyrrolidin-1-yl]acetic acid
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-(4-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
5-{4-[(2-ethylpyrimidin-4-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[3-(furan-2-yl)propyl]-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carboxamide
N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1,3-benzothiazole-5-carboxamide
1-(2-aminoethyl)-N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
4-(1H-indol-5-ylmethyl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-amino-6-cyclopropanecarbonyl-4-(5-hydroxy-2-methoxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[4-(pyrrolidin-1-yl)butyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
1-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-dihydroquinolin-4-one
2,5-dimethyl-N-(4,4,4-trifluorobutyl)pyrazolo[1,5-a]pyrimidin-7-amine
ethyl 3-({1-[4-(5-phenylpentanamido)phenyl]piperidin-4-yl}amino)propanoate
2-(3-chlorophenoxy)-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
(1S,5R)-3-benzyl-6-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
3-{[1-(2-methyl-1H-imidazole-4-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}but-3-enamide
2-methoxy-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[2-(dimethylamino)-2-(4-fluorophenyl)acetamido]cycloheptane-1-carboxamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
3-[(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)amino]propan-1-ol
(4aS,8aR)-6-(4-methylpyrimidin-2-yl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
3-[5-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
(2S,4R)-4-amino-1-[3-(cyclooctylcarbamoyl)propanoyl]-N-methylpyrrolidine-2-carboxamide
methyl 5-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-5-oxopentanoate
N-[2-(2-fluorophenyl)ethyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
1'-{3-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1,2-oxazole-5-carbonyl}spiro[indene-1,4'-piperidine]
ethyl 2-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-1,3-oxazole-4-carboxylate
3-[(dimethylamino)methyl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-ol