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(6-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)methanol
3,5-dichloro-4-methyl-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]benzamide
2-butyl-N-[2-(dimethylsulfamoyl)ethyl]-1,3-benzoxazole-5-carboxamide
1-ethyl-8-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-N-(pyridin-4-ylmethyl)-4-(pyrrolidin-3-yl)benzamide
3-{5-[2-(4-methylbenzenesulfonyl)ethyl]-1H-1,2,4-triazol-3-yl}pyridine
1-cyclopropyl-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)cyclopropanamine
2-[1-({1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]propan-2-amine
2-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-3-ol
1-tert-butyl-N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
3-({3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
6,8-dimethyl-2-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)quinolin-4-ol
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(1-hydroxybutan-2-yl)-1,3-dimethyl-2,6-dioxo-N-(pyridin-2-ylmethyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
8-[2-(2,3-dihydro-1H-isoindol-2-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(methyl){[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}amine
(isoquinolin-5-ylmethyl)(methyl){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
6-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-(3-chlorophenyl)-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]acetamide
2-methyl-5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)pyrimidin-4-ol
2-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]pyridine-3-carboxamide
7-(4-methoxy-2-methylbenzoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methoxyquinoline
8-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane
ethyl 5-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(3-phenylpropyl)-4-(pyridin-3-ylmethyl)morpholine
4-{4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}-5,6-dimethylpyrimidine
2-(4-{5-cyclopropyl-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-ol
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-6-oxo-1-propylpiperidine-3-carboxamide
2-(dimethylamino)-7-(1-methyl-1H-indole-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{2-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]pyrrolidin-1-yl}ethan-1-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-4-(2-oxopyrrolidin-1-yl)benzamide
(2S)-2-{5-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}propanoic acid
1-[6-hydroxy-4-(6-hydroxypyrimidin-4-yl)-1,4-diazepan-1-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
4-(2-ethylpyrimidine-5-carbonyl)-1-phenylpiperazin-2-one
2-chloro-N-(2-{[2-oxo-6-(propan-2-yl)-1,2-dihydropyridin-3-yl]formamido}ethyl)benzamide
6-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]-4-methylpyrimidine-5-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3,4-difluoro-N-(pyridin-3-ylmethyl)benzamide
2-(4-fluorophenyl)-2-hydroxy-N-(1H-indol-4-ylmethyl)acetamide
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-5-phenyl-1,2-oxazole-3-carboxamide
1-(2-methoxy-6-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
(4aS,7aR)-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
N-{[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
N-[5-({3-[(2-chloro-6-fluorophenyl)methyl]-1-methyl-2-oxo-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-6-yl}methyl)thiophen-2-yl]acetamide
8-[2-(3,4,5-trimethoxyphenyl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione