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4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-3-methyl-1-propyl-1H-pyrazole
3-(9H-fluoren-2-ylmethyl)-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
ethyl 4-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-amido)piperidine-1-carboxylate
(4aS,7aR)-1-(3-methyl-1,2-oxazole-5-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{3-methyl-3,9-diazaspiro[5.6]dodecane-9-carbonyl}-1,4-dihydroquinolin-4-one
3-{[(adamantan-2-yl)amino]methyl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]pyridin-2-amine
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]-2-(1H-pyrazol-1-yl)acetamide
(4aR,7aS)-1-(pyrimidin-2-yl)-4-(1H-pyrrole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-4-[({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)amino]piperidine-1-carboxamide
3-[1-(2-chloropyridine-4-carbonyl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
1-methyl-4-[2-(4H-1,2,4-triazol-4-yl)phenoxy]piperidine
2-(5-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}furan-2-yl)benzonitrile
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]propan-1-one
4-{1-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]piperidin-3-yl}benzoic acid
N,N-dimethyl-2-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}acetamide
N-[(8-methoxyquinolin-5-yl)methyl]-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
1-{3-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,3-benzotriazole
1-(4-fluoro-3-methoxybenzoyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-[3-(1-phenylcyclopropyl)-5-[3-(pyrrolidin-1-yl)propyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
(3aS,6aR)-3-[2-(piperidin-1-yl)ethyl]-5-[3-(pyridin-3-yl)propanoyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(3-{4-[(diphenylmethyl)amino]piperidin-1-yl}phenyl)pyridine-3-carboxamide
N-{1-[1-(3-cyano-2-methoxypyridin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
1-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-amino-4-cyclopropyl-6-(4-hydroxyphenyl)pyridine-3-carbonitrile
5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-2-(2,3,4-trimethoxyphenyl)pyridine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[5-methoxy-2-({[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
(3S,4S)-1-{[3-(furan-2-yl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-[1-(4-fluorophenyl)piperidin-4-yl]-4-(piperidin-1-yl)butanamide
3-cyclohexyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
N-(1-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
N-[(5,6-dimethylpyridin-3-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-[4-(benzenesulfonyl)piperazine-1-carbonyl]-1-(2-methoxyethyl)pyrrolidin-2-one
5-(1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-2-yl)-3-phenyl-1,2,4-oxadiazole
2-(3-{[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]methyl}piperidin-1-yl)ethan-1-ol
3-[(2,5-dimethylphenyl)methyl]-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-[1-(1H-indole-7-carbonyl)piperidin-4-yl]piperidin-3-ol
3-(4-{[2-(methylcarbamoyl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(3-methyl-1,2-oxazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[3-(2-phenylethyl)-1-(pyrimidin-2-yl)piperidin-3-yl]methanol
2-(methoxymethyl)-4-methyl-5-({5-[2-(methylsulfanyl)propyl]-4-phenyl-1H-imidazol-1-yl}methyl)-1,3-thiazole
ethyl 4-benzyl-1-[(4-acetamidophenyl)methyl]piperidine-4-carboxylate
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
2-(1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)ethan-1-ol
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-2-[(3-methoxyphenyl)sulfanyl]ethan-1-one
2-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-1,2-oxazinane
1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-4-(thiophen-2-yl)butan-1-one
methyl (2S,4S,5R)-1,2-dimethyl-4-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]carbamoyl}-5-phenylpyrrolidine-2-carboxylate
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-(cyclohexylmethyl)piperazin-2-one
1-[3-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-(dimethylamino)butan-1-one