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1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-methyl-5-(propan-2-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
3-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)pyridine
2-(3-{2-[2-(trifluoromethoxy)phenyl]pyridin-4-yl}pyrrolidin-1-yl)acetic acid
1-(cyclopropylmethyl)-3-(isoquinolin-5-yl)-6-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-[(2-chlorophenyl)methyl]-4-cyclopentanecarbonylmorpholine
2-(3-methyl-1,2-oxazol-5-yl)-1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
1-(2,6-dimethylpyridin-4-yl)-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
N-(4-fluoro-2-methylphenyl)-2-[2-(quinolin-2-yl)-1H-imidazol-1-yl]acetamide
N-[(3,4-difluorophenyl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
[(4-{1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidin-2-yl}phenyl)methyl]dimethylamine
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl]propanoate
ethyl 4-(8-methyl-3-{[N-(oxolan-2-ylmethyl)-1-thiophen-2-ylformamido]methyl}quinolin-2-yl)piperazine-1-carboxylate
1-cyclopentyl-3-(3-fluorophenyl)-3-{2-[4-(2-hydroxyphenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
2-methyl-4-(3-phenylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[3-(propan-2-yloxy)propyl]benzamide
N,2-dimethyl-6-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,6-dihydropyrimidine-5-carboxamide
3-[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]-2,2-dimethylpropan-1-ol
[(5-{1-cyclopentyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}thiophen-3-yl)methyl]dimethylamine
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(1H-pyrazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[7-(azepane-1-carbonyl)-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazol-5-yl]-2-cyclopentylacetamide
8-(cyclopentylmethyl)-3-[2-(4-ethylpiperazin-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-benzyl-2-[2-(2-hydroxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]acetamide
(2S)-2-amino-3-(4-hydroxyphenyl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)propanamide
1-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
4-(4-methylpyridin-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(1-ethyl-1H-pyrazol-4-yl)-7,8-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)quinoline
(3S)-3-({2-[4-(propan-2-yloxy)phenoxy]ethyl}amino)azepan-2-one
5-methyl-4-{[(2-propyl-1,3-thiazol-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
(4aR,8aR)-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-(piperidin-3-yl)benzamide
N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-3-(1,2-oxazinan-2-yl)propanamide
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
2-{1-methyl-4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperazin-2-yl}ethan-1-ol
2-[1-methyl-10-oxo-4-(propane-1-sulfonyl)-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
(3S,4S)-N-(2,3-difluorophenyl)-3-hydroxy-4-(propan-2-yloxy)pyrrolidine-1-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,2,5-oxadiazole-3-carboxamide
(3S,4R)-1-[(8-methoxyquinolin-2-yl)methyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-(3-{3-[5-(ethanesulfonyl)thiophen-2-yl]phenyl}-1H-pyrazol-1-yl)-2-methylpropan-2-ol
N-[1-(1,1-dioxo-1λ6-thian-4-yl)piperidin-4-yl]-1H-1,2,4-triazole-5-carboxamide
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)piperazin-2-one
2-ethyl-N-[4-(furan-2-yl)butan-2-yl]-4-methyl-1,3-oxazole-5-carboxamide
2-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}-6-methoxyphenol
1-benzyl-N-[1-(furan-2-ylmethyl)piperidin-4-yl]-1H-pyrazole-4-carboxamide
5-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
6-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]imidazo[2,1-b][1,3]thiazole
2-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)acetamide
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
1-[(3-fluorophenyl)methyl]-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-6-oxopiperidine-3-carboxamide