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N-benzyl-2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-ethylacetamide
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine
3-ethyl-6-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
1-[(2-chlorophenyl)methyl]-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(2-methoxyphenyl)methyl]-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]cyclopropanamine
N-cycloheptyl-N-ethyl-3-(1,2-oxazolidin-2-yl)propanamide
5-[3-(2-ethylpiperidin-1-yl)-3-oxopropyl]-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
2-[9-(1H-1,2,3-benzotriazole-5-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
2-(2,4-dimethoxyphenyl)-8-methoxy-5-[(3-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
4-[2-(4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,2,3-triazol-1-yl)ethyl]morpholine
N-(1-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-cyclopropylpyridine-2-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(pyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[4-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)thiophen-2-yl]ethan-1-one
N-{2-[(2-fluorophenyl)carbamoyl]ethyl}-N'-(2-methylphenyl)propanediamide
5-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-3-propylimidazolidine-2,4-dione
N-[(3S,4R)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-propylpyrrolidin-3-yl]methanesulfonamide
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyridine-3-carbonitrile
N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
6-methyl-2-{2-[(4-phenylbutan-2-yl)amino]ethyl}-3,4-dihydropyrimidin-4-one
ethyl 5-[(2,6-difluorophenyl)methyl]-1-[2-(dimethylamino)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-[2-(2-ethylpiperidin-1-yl)-2-oxoethyl]-3-(2-methoxyphenyl)-1-(3-methoxypropyl)pyrrolidine-2,5-dione
4-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-N-(3-hydroxyphenyl)-4-oxobutanamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]pyrazolo[1,5-a]pyridine-3-carboxamide
2-(4-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}morpholin-3-yl)acetic acid
N-[(1R,3S)-3-{[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}cyclopentyl]-1H-indazole-3-carboxamide
N-tert-butyl-3-[3-(2-hydroxyphenyl)propanamido]-2-methylbenzamide
5-(3-methoxyphenoxymethyl)-N-methyl-N-[1-(pyridin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(1-ethylpiperidine-4-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{[1-(dimethylamino)cyclohexyl]methyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
[(2S)-1-[2-(2-ethylphenoxy)ethyl]pyrrolidin-2-yl]methanol
1-[4-(benzyloxy)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-[(5-methylthiophen-2-yl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
1-(4-cyclohexyl-1,4-diazepan-1-yl)-2-(3-hydroxyphenyl)ethan-1-one
1,9-dimethyl-4-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[7-(3-methyl-4-oxopentanoyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
(3aS,6aS)-2-cyclohexyl-5-[3-(2-methyl-1H-imidazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-ethyl-1,5-dimethyl-3-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2-dihydropyridin-2-one
N-{1-[1-(3-cyclopentylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-N-methyloxolan-3-amine
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[(3-methoxyphenyl)methyl]pyrrolidin-2-one
2-(4-{[methyl(thian-4-yl)amino]methyl}phenoxy)acetic acid
4-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
{4-benzyl-1-[(3-fluorophenyl)methyl]piperidin-4-yl}methanol
5-(3-fluorophenoxymethyl)-N-(thiophen-2-ylmethyl)-1H-pyrazole-3-carboxamide
(2S,4R)-4-amino-1-{3-[(2,3-dihydro-1H-inden-5-yl)carbamoyl]propanoyl}-N-methylpyrrolidine-2-carboxamide
1'-(5-ethyl-1,3-oxazole-4-carbonyl)-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[3-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-7-methylquinolin-2-yl]piperidin-4-ol