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methyl 3-[(3S,4R)-1-[(2-ethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[3-(dimethylamino)-1-phenylpropyl]-2-(piperidin-4-yl)acetamide
5-{2-[(2,2-difluoroethyl)amino]pyrimidin-4-yl}-2-ethoxybenzoic acid
2-(dimethyl-1,3-thiazol-5-yl)-1-(7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-N-methyl-1-(2-phenylethyl)piperidin-3-amine
(3S)-1-ethyl-4-[2-(3-methoxyphenyl)-1,3-benzoxazole-6-carbonyl]-3-methylpiperazin-2-one
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-2-(morpholin-4-yl)benzamide
6-chloro-2-{6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}-1H-1,3-benzodiazole
N-(dicyclopropylmethyl)-2-(dimethylamino)-2-(4-methylphenyl)acetamide
2-(1H-1,3-benzodiazol-1-ylmethyl)-1,3-oxazole-4-carboxylic acid
2-[benzyl({[1-(propan-2-yl)-1H-imidazol-5-yl]methyl})amino]ethan-1-ol
3-(azepane-1-carbonyl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
8-(butan-2-yl)-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(trifluoromethyl)pyrimidin-2-amine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl}ethan-1-one
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}pentane-1,4-dione
4-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-2-phenylpyrimidine
2-(2,5-dioxoimidazolidin-1-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
4-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-6-(propan-2-yloxy)pyrimidin-2-amine
(3S,4S)-1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
2-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
2-{5-[1-(furan-3-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
1-methyl-2-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
3-(1,2-oxazolidin-2-yl)-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(1H-indol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methylphenyl)-3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]piperidine-4-carboxylate
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
dimethyl[(4-{1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidin-2-yl}phenyl)methyl]amine
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
methyl (2R)-2-[(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]propanoate
1-[(4-methoxyphenyl)methyl]-N-[(1R,2S)-2-phenylcyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-N-[(4-fluorophenyl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-2-oxo-2H-pyran-5-carboxamide
7-chloro-N,N-dimethyl-2-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyridine-3-carboxamide
N,N-diethyl-4-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}aniline
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
6-(1-benzothiophen-3-yl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 5-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}-5-oxopentanoate
2-{4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3-(4-methyl-1,3-thiazol-5-yl)-1-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]propan-1-one
1-[(2-fluorophenyl)methyl]-6-oxo-N-[3-(propan-2-yloxy)propyl]piperidine-3-carboxamide
methyl 5-{[(3-chlorophenyl)methyl]amino}-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3,4-dimethoxyphenyl)methyl]-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-[2-(ethylsulfanyl)ethyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-3-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}urea
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide