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2-[1-(3-phenylpropyl)-4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-methyl-2-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)acetamide
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-amino-4-{[(1R)-1-(3-methoxyphenyl)ethyl]amino}quinazoline-6-carboxylic acid
6-(2,4-difluorophenyl)-N,N-dimethylpyridine-2-carboxamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-1H-pyrazole-3-carboxamide
N-[2-(dimethylamino)ethyl]-3-{1-[1-(4-methoxyphenyl)piperidin-4-yl]piperidin-4-yl}propanamide
(1R,5S)-6-methyl-3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-(2-hydroxyphenoxy)ethan-1-one
2-{[5-(pyridin-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(pyrimidin-2-yl)morpholine
N-methyl-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}-N-(quinoxalin-6-ylmethyl)propanamide
2-{3-hexyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl}benzonitrile
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
1-[(2-methyl-1H-imidazol-4-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-[3-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]acetic acid
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-cyclobutyl-1,3-oxazole-4-carboxamide
N,N-diethyl-2-{4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
N-{1-[4-(4-methoxyphenyl)-3-oxopiperazin-1-yl]-1-oxopentan-2-yl}acetamide
3-{5-[(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1H-1,2,4-triazol-3-yl}pyridine
2-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)-8-benzyl-2,8-diazaspiro[5.5]undecane
{3-[(4-fluorophenyl)methyl]-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-3-yl}methanol
(3S,4R)-4-(4-fluorophenyl)-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)pyrrolidine-3-carboxylic acid
N-(3-methyl-1-{7-[(3,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
3-(5-acetyl-2-ethoxyphenyl)-1-[2-(morpholin-4-yl)ethyl]urea
2-butyl-N-(3,4-dimethoxyphenyl)-2,5-dihydro-1H-pyrrole-1-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
6-ethyl-2-methyl-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]quinoline-4-carboxamide
1-(2-cyclopentylacetyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
(3R,4S)-1-(benzenesulfonyl)-4-propylpyrrolidin-3-amine
N,N,4,5-tetramethyl-6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidin-2-amine
1-(1H-imidazol-2-ylmethyl)-4-(2-methylphenoxy)piperidine
(4aS,7aR)-1-(4-methyl-1H-imidazole-5-carbonyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
1-benzyl-8-cyclopentyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
2,3-difluoro-5-(1H-imidazol-1-yl)phenol
4-fluoro-N-{2-[(3-methyl-4-oxo-3,4-dihydroquinazolin-7-yl)formamido]ethyl}benzamide
methyl 5-{[(4-ethylphenyl)methyl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(3,4-dichlorophenyl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-propoxyethan-1-one
2-({3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-6-methoxyphenol
N-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
N-methyl-2-(4-methyl-1,4-diazepan-1-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
3-({[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]carbamoyl}amino)-N,2-dimethylbenzamide
1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-4-(piperidin-1-yl)butan-1-one
N-(cyclopropylmethyl)-5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl({[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}){[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
3-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide