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5-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]-4-methyl-2-(pyridin-3-yl)pyrimidine
N-[1-(methoxymethyl)cyclopentyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-methyl-11-{[2-(trifluoromethyl)phenyl]methyl}-3,7,11-triazaspiro[5.6]dodecane
1-(furan-2-carbonyl)-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
(2S,4S)-4-amino-N-(propan-2-yl)-1-(quinolin-2-ylmethyl)pyrrolidine-2-carboxamide
1-(1H-imidazol-2-ylmethyl)-4-(2-methylphenyl)-1,4-diazepane
3-({[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
3-{[1-(3,4-dimethylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
N-[3-(2-methoxyphenyl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
8-(3,5-difluoropyridine-2-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
7-methyl-2-{2-[5-oxo-2-(thiophen-2-yl)cyclopent-1-en-1-yl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
1-[(3-chlorophenyl)methyl]-N-{[1-(2-phenylethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]urea
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(oxolan-3-yl)acetamide
1-methyl-4-[(1-propyl-1H-imidazol-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(oxan-4-yl)acetamide
N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
1-{4-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1'-(3,6-dimethylpyrazin-2-yl)-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}pyrrolidin-2-one
3-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}piperidine-1-carboxamide
3-cyclohexyl-N-(1,2-oxazol-3-ylmethyl)-1H-pyrazole-4-carboxamide
1-[(2-methylphenyl)methyl]-N-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-(4-ethoxyphenyl)-N-(thiophen-3-ylmethyl)acetamide
2-(2-hydroxyethyl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
1-cyclopentyl-4-[4-(pyridin-3-yl)pyrimidin-2-yl]piperazin-2-one
1-[2-(4-benzylpiperazin-1-yl)ethyl]-3-(2-chloropyridin-3-yl)urea
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-3-(2-fluorophenoxymethyl)piperidine
dimethyl({[(3R,4S)-4-(propan-2-yl)-1-(pyrimidin-2-ylmethyl)pyrrolidin-3-yl]sulfamoyl})amine
3-(adamantane-1-carbonyl)-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[2-(4-fluorophenyl)morpholin-4-yl]quinoline-4-carboxylic acid
N-methyl-3-(1,2-oxazinane-2-carbonyl)pyridin-2-amine
3,5-dimethyl-4-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
5-fluoro-2-{3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propyl}-1H-1,3-benzodiazole
N-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-2-(pyridin-2-yl)pyrrolidine-1-carboxamide
7-(3,6-dimethylpyrazin-2-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
(2R,3S,6R)-5-(6-ethylpyrimidin-4-yl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
ethyl (4aS,8aR)-6-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-decahydro-1,6-naphthyridine-4a-carboxylate
7-(3-chlorophenyl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-ethyl-5-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
5-[3-methyl-5-(phenoxymethyl)furan-2-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
8-{[2-(ethylamino)pyrimidin-5-yl]methyl}-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-(4-methoxy-3,5-dimethylphenyl)acetic acid
N-methyl-N-[(5-methylfuran-2-yl)methyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
propyl 4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide