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2-{1-[(1-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}benzoic acid
1-cyclobutanecarbonyl-N-[2-hydroxy-2-(3-methoxyphenyl)ethyl]piperidine-4-carboxamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-3-yl]propanamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carboxylic acid
3-ethyl-1-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)urea
7-(2-ethoxybenzoyl)-N-(prop-2-en-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-4-(4-methoxybenzoyl)piperazine
6-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-N-[(2-fluorophenyl)methyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
4-[1-(4-chlorophenyl)cyclohexanecarbonyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
methyl 1-[(3S,5S)-1-[(4-methoxy-3-methylphenyl)methyl]-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-cyclopentyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carboxamide
N-({1-[2-(carbamoylamino)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-N-methylcyclohexanecarboxamide
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]isoquinoline
N-{1-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-2-(methylamino)acetamide
3-(1-{1-[(2S)-2-amino-3-hydroxypropanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
N-[(2R,3R)-2-methoxy-1'-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
N-[(1S,2R)-2-[(1-acetylpiperidin-4-yl)amino]cyclobutyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
6-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl}-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
8-fluoro-2-{[(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amino]methyl}quinolin-4-ol
N,N-dimethyl-5-[8-methyl-4-(2-methylpiperidine-1-carbonyl)quinolin-2-yl]pyrimidin-2-amine
N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-(2-methoxybenzoyl)-4-{[1,2,4]triazolo[4,3-a]pyridine-7-carbonyl}piperazine
2-methoxy-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methylpropanamide
4-({5-[2-chloro-4-(4H-1,2,4-triazol-4-yl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
1-(1H-1,2,3-benzotriazol-5-yl)-3-[2-(dimethylamino)ethyl]-3-ethylurea
{1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
2-methoxy-N-({8-[(2,3,6-trifluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
5-chloro-2-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline
(3-{2-[1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-{5-[4-(aminomethyl)phenyl]-3-(3,4-difluorophenyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-phenoxyacetamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
6-({[1-(6-chloro-1,3-benzothiazol-2-yl)piperidin-4-yl]amino}methyl)pyrimidin-4-ol
2-[(4aS,7aR)-6,6-dioxo-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoacetamide
1,3-dimethyl-5-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
8-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-3-ol
2-(2,3-dimethoxyphenyl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
1-(azocan-1-yl)-3-(2-methoxy-4-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-[4-(methylsulfanyl)benzoyl]piperidine
1-(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepane
(1S,3R)-N1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
(1S,5R)-6-(3,5-dimethylbenzoyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(5-methoxy-2-{[(3-methylbutyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
N-cycloheptyl-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
5-(1-{[4-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-3-[2-(4-methoxyphenyl)ethyl]-5-methylimidazolidine-2,4-dione
{3-[(4-fluorophenyl)methyl]-1-[3-(methylsulfanyl)propyl]piperidin-3-yl}methanol
methyl 3-chloro-4-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]amino}benzoate