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(2S,4R)-4-amino-N-ethyl-1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidine-2-carboxamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-(3,4-difluorobenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[7-(1-benzofuran-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1-phenylmethanesulfonamide
1-(2-{[2-(furan-2-yl)-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)imidazolidin-2-one
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)(2-phenylethyl)amine
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}amine
(1H-1,3-benzodiazol-2-ylmethyl)[(2-fluorophenyl)methyl](2-methoxyethyl)amine
2-(adamantan-1-yl)-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)acetamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-1-methyl-N-(2-methylpropyl)-1H-imidazole-2-carboxamide
5-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1'-methyl-3,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[(2R,3R,6R)-5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-[(4-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-3-methoxyphenyl)methyl]-1λ6-thiomorpholine-1,1-dione
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[2-(2-phenylethyl)morpholin-4-yl]ethan-1-one
4-{3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-4H-1,2,4-triazole
N-[2-(1H-indol-3-yl)ethyl]-3-methyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-5-carboxamide
(1S,5R)-3-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetyl)-3,9-diazabicyclo[3.3.2]decan-10-one
3-fluoro-N-methyl-N-[2-(pyridin-4-yl)ethyl]pyridine-4-carboxamide
6-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
3-[2-(2,4-difluorophenyl)ethyl]-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine
2-(5-fluoro-2-methoxyphenyl)-2-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}acetic acid
N-methyl-N-(4-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]acetamido}phenyl)acetamide
N-ethyl-2-{4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-4-carboxamide
1-(2-methylpropyl)-5-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]pyrrolidine-3-carboxamide
4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
4-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-5-propylpyrimidine
N-(2-hydroxyethyl)-4-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-5-carboxamide
N-ethyl-4-hydroxy-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N-butyl-N-ethyl-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2R)-2-amino-4-methyl-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pentan-1-one
4-benzyl-1-[2-(4-methanesulfonylpiperazin-1-yl)-2-oxoethyl]pyrrolidin-2-one
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-(pyrrolidine-3-carbonyl)piperidine
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}cyclobutanecarboxamide
(1S,5R)-6-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-cycloheptyl-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
3-{4-phenyl-5-[4-(pyrimidin-5-yl)phenyl]-1H-imidazol-1-yl}propan-1-ol
2-cyclopropyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyrimidine-5-carboxamide
N-[1-({5-[3-(1H-pyrrol-1-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)pyrrolidin-3-yl]acetamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]imidazo[1,2-a]pyridine-2-carboxamide
4-methyl-N-(2-{7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
3-methyl-N-[(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-3-yl)methyl]but-2-enamide
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-5-(2-methylphenyl)-1,2,4-triazin-3-amine
2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]morpholin-3-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-cyclopentyl-4-{[methyl({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amino]methyl}pyrrolidin-2-one
(3S,4R)-1-[4-(difluoromethoxy)benzenesulfonyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
4-{1-[(3-fluorophenyl)methyl]piperidin-3-yl}-5-phenyl-2-(pyridin-4-yl)pyrimidine
1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidine-3-carboxamide
3-[(cyclohex-3-en-1-ylmethyl)amino]-N-[2-(1H-imidazol-1-yl)ethyl]-5-(pyrrolidine-1-sulfonyl)benzamide
1-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-1,2,3,4-tetrahydroquinolin-2-one