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1-(furan-2-carbonyl)-4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazine
2-[1-methyl-10-oxo-4-(pyrimidin-2-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
5-({9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
1-(cyclopentylmethyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(2-methoxyphenyl)methyl]piperidin-4-ol
{[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
N-cyclopentyl-N-[(2,5-dimethoxyphenyl)methyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 4-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-amido]piperidine-1-carboxylate
1-[2-methoxy-5-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
(1S,6R)-9-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
3-{1-[(6-ethoxyquinolin-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
3-(1-hydroxy-3-methylbutan-2-yl)-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
5-tert-butyl-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1,3,4-oxadiazol-2-amine
(3R,4R)-4-amino-1-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}piperidin-3-ol
1-(4-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N'-(2-chlorophenyl)-N-[(1-methylpyrrolidin-3-yl)methyl]ethanediamide
1-{5-[3-(4-methoxy-2-methylbenzoyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(2,5-dimethylphenoxy)-N-methylpropanamide
(1R,5R)-N-(3-fluorophenyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N'-(2-ethoxyphenyl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanediamide
methyl 1-benzyl-3-cyclopropaneamido-5-[(3-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N,N-dimethyl-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrazine-2-carboxamide
N,N-diethyl-1-({1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
(3S)-4-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
1-(2-{2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}propyl)-1H-1,2,4-triazole
5-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-propylpiperidin-2-one
(3S,4R)-3-benzyl-1-(1H-indole-2-carbonyl)-4-methylpiperidin-4-ol
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[2-(diethylamino)ethyl]-5-(methoxymethyl)-N-methyl-1H-pyrazole-4-carboxamide
[(3R,5S)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-8-fluoro-N-methylquinoline-2-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(6-hydroxypyrimidin-4-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
3-(2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
2-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-2H-1,2,3-benzotriazole
4-[(4-fluorophenyl)methyl]-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
2-{3-cyclopentyl-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazol-1-yl}benzoic acid
2-({4H,5H,6H,7H,8H-cyclohepta[b]thiophen-2-ylmethyl}[(1-methyl-1H-imidazol-2-yl)methyl]amino)ethan-1-ol
N,5-dimethyl-2-phenyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}furan-3-carboxamide
[(3R,4R)-1-(2,5-difluorobenzoyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
2-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
1-[4-(2-methylphenoxy)piperidin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
2-[5-(5-methyl-2H-1,2,3-triazol-4-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-{3-oxo-3-[2-(3-phenylpropyl)morpholin-4-yl]propyl}pyrrolidin-2-one
2-(2-hydroxyethyl)-8-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-2,8-diazaspiro[5.5]undecan-3-one