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N-[(3-methoxyphenyl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
1-(furan-2-ylmethyl)-4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}piperidine
6-[(3aS,6aR)-2-oxo-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-(9H-purin-6-yl)piperidin-4-amine
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-1-methyl-1H-indole-3-carboxamide
1-[(2-chlorophenyl)methyl]-N-(2-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2,3-dihydro-1H-indene-1-carboxamide
2-[(3R,4S)-3-(2-methoxy-2-methylpropanamido)-4-(propan-2-yl)pyrrolidin-1-yl]pyridine-3-carboxamide
4-methoxy-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)benzamide
2-(4-fluorobenzoyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,5,6-trimethylpyrimidin-4-amine
(2S)-1-[(3-chloro-4,5-dimethoxyphenyl)methyl]-2-(methoxymethyl)pyrrolidine
3-chloro-N-(4-{4-[(furan-2-ylmethyl)amino]piperidin-1-yl}phenyl)benzamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
4-chloro-2-{[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenol
ethyl 4-{[2-(2-fluorophenoxy)phenyl]carbamoyl}piperazine-1-carboxylate
4-[(2S)-2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-6-fluoro-1,2-dihydroquinolin-2-one
N-(3,5-dimethoxyphenyl)-2-{[1-(1H-1,2,4-triazol-5-yl)ethyl]amino}acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-(morpholin-4-yl)benzamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}pyridine-3-sulfonamide
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
2-({1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)benzonitrile
3-[2-(2,6-difluorophenyl)ethyl]-1-(1,3-thiazol-4-ylmethyl)piperidine
N3-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-N5-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-N-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}benzamide
5-(2-methylpropanoyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(4-methoxyphenyl)methyl]morpholine
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-1H-imidazole-2-carboxamide
5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-1-[2-(1H-imidazol-5-yl)ethyl]-3-methyl-1H-1,2,4-triazole
(4aR,8aR)-2-(2-methyl-1H-pyrrole-3-carbonyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
3-(3-hydroxy-3-methylbutyl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]benzamide
5-(4-acetyl-2-methoxyphenoxymethyl)-N-[2-(piperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
5-chloro-N-methyl-6-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,6-dihydropyridine-3-carboxamide
4-[4-(4-methylphenyl)-2-[(oxan-4-yl)amino]pyrimidin-5-yl]phenol
3-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-methyl-1-(4-phenoxyphenyl)urea
1-[2-(1-benzothiophen-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(prop-2-en-1-yl)piperidine-3-carboxamide
N-[2-(dimethylamino)ethyl]-3,4-dimethoxy-N-{[8-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}benzamide
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl][(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]methylamine
(1R,3S)-7-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-7-azaspiro[3.5]nonane-1,3-diol
2-[4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
(1R,5S)-3-[4-(4-chlorophenoxy)piperidine-4-carbonyl]-3,8-diazabicyclo[3.2.1]octane
3-[4-(2-ethoxyethyl)piperazine-1-carbonyl]-5,6,7,8-tetrahydroquinoline
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}but-3-en-1-one
methyl({[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})(pyridin-2-ylmethyl)amine
5-(2-chloro-6-fluoro-3-methylbenzoyl)-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-cyclobutyl-2-(2-phenylethyl)morpholine