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2-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,3-thiazole-4-carboxamide
3-[(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]benzonitrile
N,N-bis(propan-2-yl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carboxamide
N-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-3-yl]methyl}-3-(trifluoromethyl)benzamide
1-cyclobutyl-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
6-(2-chlorophenyl)-N-[(2S)-1-hydroxypropan-2-yl]-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidine
1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
(3R,7S,8aS)-7-{[(4-methoxyphenyl)methyl]amino}-3-(2-methylpropyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[2-(4-cyclopropanecarbonylphenyl)ethyl]pyrrolidin-2-one
3-benzyl-5-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazole
ethyl 1-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-4-(2-phenylethyl)piperidine-4-carboxylate
N-cyclopropyl-1-[5-(hydroxymethyl)furan-2-carbonyl]piperazine-2-carboxamide
3,5-dimethyl-N-{3-methyl-1-[7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}benzamide
5-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole
N'-(2,4-dimethylphenyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]propanediamide
4-(benzyloxy)-1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
1-(1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperidin-4-yl)-2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
methyl 3-[(3S,4R)-4-(morpholin-4-yl)-1-[(4-oxo-4H-chromen-3-yl)methyl]piperidin-3-yl]propanoate
(2-{[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]methyl}phenyl)methanol
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
1-(2-{1-[6-(cyclopentylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(4-ethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2-fluorophenyl)methyl]-3-{1-[3-(2-oxopiperidin-1-yl)propanoyl]piperidin-3-yl}propanamide
2-methyl-4-{4-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-[(5-ethylpyridin-2-yl)methyl]-N-methylpropanamide
N-(1-hydroxy-2-methylpropan-2-yl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-{[(3-aminopropyl)amino]methyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
(1R,5S,6R,7S)-3-(2-aminoethyl)-4-oxo-N-[2-(thiophen-2-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
N-[5-({1-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)thiophen-2-yl]acetamide
2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methylacetamide
2-(3-fluorophenyl)-2-[2-(2-methyl-1,3-thiazol-4-yl)acetamido]acetic acid
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
2-[1-(propan-2-yl)-5-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-3-yl]pyridine
N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-4-carboxamide
5-ethyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,3,4-oxadiazol-2-amine
N-[(1S)-1-cyclohexyl-2-hydroxyethyl]-4-(1H-pyrazol-4-yl)butanamide
3-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}urea
1-[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]-2-(quinazolin-4-yloxy)ethan-1-one
4-(4-fluorophenoxy)-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]piperidine
3-[(3R,4S)-4-(dimethylamino)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl]propanoic acid
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[2-(methylsulfanyl)phenyl]methyl}amine
1-{4-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
2-[(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-4,6-dimethylpyridine-3-carbonitrile
1-{2-[(5-methyl-2-phenylfuran-3-yl)formamido]ethyl}piperidine-3-carboxamide
8-methyl-N-[2-(5-methylfuran-2-yl)ethyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
2-amino-N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-4-methylpyrimidine-5-carboxamide