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5-[(3S,4R)-4-amino-3-methoxypiperidine-1-carbonyl]-N-phenylpyrimidin-2-amine
N-methyl-2-(1-methyl-1H-imidazol-2-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-(4-methoxy-2-methylbenzoyl)piperidine
8-(4-phenylbutan-2-yl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-(butan-2-yl)phenyl]-2-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]acetamide
8-[2-(2-chloro-4-fluorophenyl)acetyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-[3-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-5-[1-(3-phenylpropyl)piperidin-4-yl]imidazolidine-2,4-dione
5-{1-[(3-chlorophenyl)methyl]-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1,2-dimethyl-1H-imidazole
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}[(2-methoxyphenyl)methyl]methylamine
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
[(3aS,6aS)-2-[4-(piperidin-1-ylmethyl)benzoyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
N-(1-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylpyridine-2-carboxamide
3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-{4-[2-(pyridin-2-yl)ethoxy]phenyl}urea
(3S,5R,9R)-5-hydroxy-11-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-[5-cyclobutyl-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-phenoxypropan-1-one
9-(cyclopropylmethyl)-1-methyl-4-(1-methyl-1H-pyrazole-4-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}-2-[4-(propan-2-yl)phenyl]acetic acid
(2S)-2-({2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)propanamide
N-(4-{[ethyl(oxan-4-ylmethyl)carbamoyl]methoxy}phenyl)propanamide
2-(3-methylbut-2-en-1-yl)-8-[2-(thiophen-2-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
dimethyl[(6-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrazin-2-yl)methyl]amine
2-(4-methyl-1,4-diazepan-1-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]acetamide
N,N-diethyl-2-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-1,2,3-triazol-1-yl)acetamide
(3R,9aR)-8-(3-chlorobenzoyl)-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-methyl-2-oxo-8-(2-phenylethyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
9-(2-methyl-6-propylpyrimidin-4-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{2-methyl-1-[2-(pyridin-2-yl)piperidin-1-yl]propan-2-yl}morpholine
(3aS,6aS)-2-(cyclopropylmethyl)-5-(1,3-dihydroxypropan-2-yl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
4-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-2,3-dihydro-1H-imidazol-2-one
N-methyl-6-(2-methylphenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-2-(thiophen-2-yl)acetamide
1-(furan-2-ylmethyl)-N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]piperidine-4-carboxamide
3-{[(carbamoylmethyl)(methyl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2,6-diamino-4-[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N-cyclopentyl-2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carboxamide
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]pyrimidin-4-amine
8-(1-methylcyclopropanecarbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3,5-dimethyl-N-{3-methyl-1-[7-(3-methylbut-2-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}benzamide
2-methyl-7-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2,7-diazaspiro[4.5]decane
2-({3-[(2R,6R)-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]phenyl}amino)acetic acid
1-(4-{[cyclopropyl(ethyl)amino]methyl}-2-methoxyphenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
2-methyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}thieno[3,2-d]pyrimidin-4-amine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-1-yl)acetamide
5-methyl-2-(4-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}piperidin-4-yl)pyridine
4-(3-ethoxyphenoxymethyl)-2-(furan-2-yl)-5-methyl-1,3-oxazole