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9-(2-phenoxyacetyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-6-[(oxolan-2-ylmethyl)amino]-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
methyl (2R,4S)-4-hydroxy-1-[(6-methoxypyridin-3-yl)methyl]piperidine-2-carboxylate
1-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-[3-(1H-indol-1-yl)propyl]-1-methylpiperidine-2-carboxamide
5-{2-[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}-1-methylpiperidin-2-one
3-{methyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amino}-1-phenylpropan-1-ol
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(2-oxoazepan-1-yl)acetamide
1-{4-[({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]piperidin-1-yl}ethan-1-one
6-({1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}amino)pyridine-3-carbonitrile
4-cyclobutaneamido-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
1-{[1,2,4]triazolo[4,3-a]pyridine-7-carbonyl}piperidin-3-amine
5-{2-[4-(4-methylpiperazin-1-yl)phenyl]-1H-imidazol-1-yl}-1H-1,2,3-benzotriazole
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(2-phenoxyethyl)-1H-pyrazole-3-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-[2-(phenylsulfanyl)acetyl]pyrrolidine-2-carboxamide
(2R,6R)-1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
2-{9-[(3-methylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
(1S,5R)-N-(4-chloro-2-methylphenyl)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[3-(pyridin-3-yl)azetidin-1-yl]-4-(trifluoromethyl)pyridine
1-(1-benzofuran-2-ylmethyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
3-({[3-(4-fluorophenoxy)propyl](methyl)amino}methyl)-N-methylpyridin-2-amine
2-(4-{[1-(propan-2-yl)-1H-indol-3-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
5-{[4-(2-methoxybenzoyl)piperazin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
4-(2,2-dimethyloxan-4-yl)-1-[(5-methyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazole
1-[2-(butan-2-yloxy)phenyl]-3-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}urea
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-hydroxy-2-(4-methoxyphenyl)acetamide
3-({[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}methyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
2-[(1-hydroxypropan-2-yl)amino]-N-(2,3,4-trifluorophenyl)acetamide
5-{1-benzyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-1-methyl-1,2-dihydropyridin-2-one
methyl(2-phenoxyethyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
(5S,9aS,9bS)-2-methyl-5-(2,4,5-trimethylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(2H-1,3-benzodioxol-5-yl)-6,8-dioxo-2,7-diazaspiro[4.4]nonane-2-carboxamide
1-ethyl-3-[(3S)-3-ethylmorpholine-4-carbonyl]-6,7,8-trifluoro-1,4-dihydroquinolin-4-one
8-(6-aminopyridine-3-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-{4-fluoro-3-[({[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}carbamoyl)amino]phenyl}propanamide
4-(3,4-dimethoxybenzoyl)piperazine-2-carboxylic acid
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2,3-dihydro-1-benzothiophene-2-carboxamide
8-[(4-methanesulfonylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
8-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2,2-difluoroethyl)-4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4-[(2,4-dimethoxy-3-methylphenyl)methyl]-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
ethyl 4-(3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperazine-1-carboxylate
2-cyclopentyl-N-[2-(1,3-thiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(1-aminocyclopropanecarbonyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
2-methyl-5-{[4-(4-propylpiperazine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}-1,3-benzothiazole
2-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
5-(2,4-difluorophenoxymethyl)-N-ethyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
N-[2-(morpholin-4-yl)ethyl]-3-azaspiro[5.5]undecan-9-amine