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4-[3-(oxolan-3-yl)-5-[2-(4,5,6,7-tetrahydro-1H-indazol-3-yl)ethyl]-1H-1,2,4-triazol-1-yl]benzonitrile
(2S,4R)-4-amino-N-(propan-2-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidine-2-carboxamide
N-(pyridin-2-ylmethyl)-1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazole
5-(2-ethoxypyridin-3-yl)-2-fluorobenzamide
3-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-indazole
1-{2-[2-amino-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
2-{4-[(2-fluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(dimethylamino)-2-(3-fluorophenyl)-N-{1-[(4-methylphenyl)methyl]cyclopropyl}acetamide
5-methyl-1'-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3aR,5S,6S,7aS)-2-(3-fluoro-2-methoxybenzoyl)-octahydro-1H-isoindole-5,6-diol
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(4-methoxyphenoxy)piperidine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-hydroxy-1-methylpiperidine-4-carbonyl)pyrrolidine-3-carboxylic acid
2-[3-(2-methoxyethyl)-5-[1-(morpholin-4-yl)propan-2-yl]-1H-1,2,4-triazol-1-yl]benzoic acid
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
5-fluoro-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1H-indole
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-(5-methylfuran-2-yl)benzamide
1-methyl-3-[3-(pyridin-4-yl)propyl]-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-chloro-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-2-methylpropanamide
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-[(2-methylphenyl)sulfanyl]acetamide
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
4-benzyl-3-ethyl-1-[2-(3-hydroxyphenyl)acetyl]-1,4-diazepan-5-one
6-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-2-methylpyrimidin-4-ol
4-(2,6-dimethylpyridin-3-yl)-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidin-2-amine
1-[3-(1H-pyrazol-1-yl)propyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
(1S,5R)-6-(1H-indol-5-ylmethyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)quinoline
5-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}furan-2-yl)-3,4-dimethyl-1,2-oxazole
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-1H-pyrazole-3-carboxamide
5-chloro-2-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenol
8-(5-chloro-3-fluoropyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(3,4-dichlorophenoxy)-1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}ethan-1-one
3-fluoro-4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-(pyridin-4-yl)quinoline
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
methyl 4-{[3-(1H-indol-2-yl)phenyl]carbamoyl}piperidine-1-carboxylate
2-(2,6-difluorophenyl)-1-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
2-[(2-{4-[(dimethylamino)methyl]phenyl}pyrrolidin-1-yl)methyl]benzoic acid
N-(2,3-dihydroxypropyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-[3-(hydroxymethyl)phenyl]-2-[methyl({[1-(morpholin-4-yl)cyclohexyl]methyl})amino]acetic acid
(1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)methanol
methyl 5-{[(2,4-dimethoxyphenyl)methyl]amino}-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[1-(4-methylphenyl)cyclopropanecarbonyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-methyl-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[4-(furan-2-ylmethyl)piperazin-1-yl]pyrimidine-5-carboxylic acid
2-[methyl(1-methylpiperidin-4-yl)amino]-1-[4-(3-methylphenoxy)piperidin-1-yl]ethan-1-one
1-(2-{[(2-chloro-6-fluorophenyl)methyl]amino}ethyl)-N-(thiophen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide