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1-methoxy-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,8-diazaspiro[4.5]decan-2-one
N'-(2-ethoxyphenyl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methylpropanediamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(thiophen-3-yl)acetamide
5-{1-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-4-phenyl-1H-imidazol-5-yl}-2-methoxyphenol
(4aS,8aR)-6-(pyrazine-2-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-cyclopropyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]quinoxaline-5-carboxamide
1'-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1,2-dihydroquinolin-2-one
5-(3-fluorophenoxymethyl)-N-[(3R)-4-hydroxy-3-methylbutyl]-1H-pyrazole-3-carboxamide
3-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide
1-ethyl-3-{1-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-imidazol-2-yl}piperidine
2-({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}amino)pyridine-3-carboxamide
methyl[(4-methylphenyl)methyl]{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
3-ethyl-1-(2-phenylethyl)-8-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(8-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)formamido]-N-(propan-2-yl)acetamide
[(6-methoxypyridin-3-yl)methyl](methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
4-[(5-{thieno[2,3-d]pyrimidin-4-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]thiomorpholine
(3S,5R)-3-(3-fluorophenoxymethyl)-1-(2-methylpropyl)-5-(pyrrolidine-1-carbonyl)piperidine
methyl({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})[(5-propyl-1H-pyrazol-3-yl)methyl]amine
3-(2-methyl-1,3-benzothiazol-5-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-3-yl]urea
2-(2-{[(4aS,7aR)-4-(cyclopropylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}phenoxy)acetic acid
8-cyclopropanecarbonyl-2-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(1H-indazol-3-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(2-methylphenyl)-N-(propan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[1-(pyrimidin-2-yl)piperidin-3-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
(3S,4R)-3-methoxy-1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-amine
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-5-phenoxyfuran-2-carboxamide
2-(4-methyl-1,4-diazepan-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
5-methanesulfonyl-2-methyl-4-[3-(pyridine-3-carbonyl)piperidin-1-yl]pyrimidine
4-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)pyrimidine
N-(isoquinolin-5-ylmethyl)-N,3,5-trimethyl-1-benzofuran-2-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-(1H-imidazol-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-{1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]azetidin-3-yl}pyridine
2-(3,4-dimethoxyphenyl)-2-{methyl[2-(morpholin-4-yl)ethyl]amino}acetic acid
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-5-methyl-1,2-oxazole-4-carboxamide
3-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-N'-cycloheptylbutanediamide
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-(thiophene-3-carbonyl)-1,4-diazepan-6-yl]oxy}acetamide
4-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-(1-methylpiperidin-4-yl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-[2-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-2-yl)ethyl]phenol
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(pyridin-4-ylsulfanyl)acetamide
1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(5-methylfuran-2-yl)-1H-imidazole
(2S,4R)-4-(dimethylamino)-1-[(2-hydroxy-6-methoxyphenyl)methyl]pyrrolidine-2-carboxylic acid
3-methyl-5-({3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1,2-benzoxazole
3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-(3-ethylphenyl)urea
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-(3-phenoxypropanoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
2-[4-(2-cyanophenyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide