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2-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carbonyl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
5-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl][(6-fluoroquinolin-2-yl)methyl](pyridin-3-ylmethyl)amine
6-ethyl-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3R,9aR)-3-(hydroxymethyl)-8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{4-[(1-cyclopropylethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(pyridin-3-yl)ethan-1-one
4-({2-[2-(furan-2-yl)phenyl]-1H-imidazol-1-yl}methyl)benzene-1-sulfonamide
N-(1,4-dioxan-2-ylmethyl)-4-(3-hydroxy-3-methylbutyl)benzamide
2-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)pyridine
5-({[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amino}methyl)pyrrolidin-2-one
3-(3-chloro-1,2-oxazol-5-yl)-1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)propan-1-one
N-[(3S,5S)-1-cycloheptyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-5-methyl-1,2-oxazole-3-carboxamide
1-(3-methylpyrazin-2-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-N,2-dimethyl-4-phenylpyridine-3-carboxamide
N-methyl-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)benzamide
4-(1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-4-carbonyl)morpholine
N-(4-methoxyphenyl)-1-(pyridine-3-carbonyl)piperidin-3-amine
2,4-dimethyl-N-{1-[4-({2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}carbamoyl)phenyl]-1H-pyrazol-4-yl}benzamide
1-ethyl-6-methyl-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydropyridin-2-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,2,2-trimethylpropanamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-(2,3-dimethylphenyl)piperidin-4-amine
N-[(3R,4S)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-propylpyrrolidin-3-yl]cyclobutanecarboxamide
2-[4-(propan-2-yl)benzenesulfonyl]-2,7-diazaspiro[4.5]decane
N-[(3R,4R)-3-hydroxy-1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]pyridine-2-carboxamide
N-[1-(1H-indol-5-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-[methyl(pyrazin-2-ylmethyl)amino]-2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}acetic acid
5-{[3-(3-chlorophenyl)pyrrolidin-1-yl]methyl}-3-(cyclopropylmethyl)-1,2,4-oxadiazole
N-[1-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)piperidin-4-yl]pyrimidin-2-amine
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
N-{[3-methyl-7-(3-methylfuran-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
7-(1-benzothiophen-3-yl)-9-hydroxy-N,N-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-sulfonamide
ethyl 2-{1-[5-(cyclooctylcarbamoyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridin-3-yl]-N-methylformamido}acetate
5-methyl-2-[4-(thiomorpholin-4-ylmethyl)phenyl]-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
N-[2-(4-methoxyphenyl)phenyl]-1-(prop-2-ene-1-sulfonyl)pyrrolidine-2-carboxamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(1H-pyrrole-2-carbonyl)-1,4-diazepan-5-one
2-[3-oxo-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-8-yl]acetic acid
N-(propan-2-yl)-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-cyclopropylacetamide
1-[(1,4-dimethyl-1H-pyrazol-5-yl)methyl]-4-(pyrrolidin-1-yl)piperidine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-1-methylazepane-2-carboxamide
1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-N-phenylpiperidin-3-amine
(2E)-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-3-(thiophen-2-yl)prop-2-enamide
4-amino-1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
2-amino-6-(6-methoxypyridin-3-yl)-4-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
N-[(1R)-1-(3-methoxyphenyl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
8-chloro-2-({4-cyclopropyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)quinoline
N-[2-(7-{[3-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclobutanecarboxamide
methyl 5-{[(2-fluoro-5-methoxyphenyl)methyl]amino}-1-methyl-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-hydroxy-1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one