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5-amino-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-1H-pyrazole-3-carboxamide
6-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidine-1-carbonyl]-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
7-fluoro-2-methyl-N-[1-(thian-4-yl)piperidin-4-yl]quinoline-4-carboxamide
2-[3-(2-methoxyethyl)-5-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,4-triazol-1-yl]pyridine
3-{[1-(2-{imidazo[1,2-a]pyridin-3-yl}acetyl)pyrrolidin-3-yl]methyl}benzamide
2-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-N-methylpyrimidin-4-amine
3-{[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]formamido}-N-phenylpropanamide
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl){[3-(pyridin-2-ylmethoxy)phenyl]methyl}amine
N-cyclopentyl-3-{[2-(pyridin-2-yl)ethyl]sulfamoyl}benzamide
4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N5-(2-methoxyethyl)-N3-methyl-1-(3-methylbutyl)-N3-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
4-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-3-yl]benzoic acid
{[(1R,5S,6R)-3-(dimethyl-1,2-oxazole-4-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]methylamine
2-({[1-(cyclopropylmethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)acetamide
ethyl 4-[1-(naphthalen-1-ylmethyl)piperidin-3-yl]piperazine-1-carboxylate
N-(3-methoxypropyl)-6-[(2S)-4-methyl-2-phenylpiperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-(dimethylamino)-N-[2-methyl-5-({[1-(3-methylpyridin-2-yl)propan-2-yl]carbamoyl}amino)phenyl]acetamide
4-[(2,4-dimethoxyphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
1-(4-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1H-pyrazol-3-yl)-1H-1,2,3,4-tetrazole
2-{2-methyl-3-[({[2-(1H-pyrazol-1-yl)phenyl]methyl}amino)methyl]-1H-indol-1-yl}acetamide
ethyl 1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxylate
2-{4-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]piperazin-1-yl}-1-(pyrrolidin-1-yl)ethan-1-one
1-(cyclohex-3-ene-1-carbonyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
2-methoxy-2-phenyl-N-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
(4aR,8aR)-2-methanesulfonyl-7-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(dimethyl-1,2-oxazol-4-yl)acetamide
N-{[7-chloro-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)furan-3-carboxamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazine
5-{[2-(2-aminoethyl)morpholin-4-yl]methyl}-2-methoxyphenol
N-(1-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-cyclopropylpyridine-2-carboxamide
1-[6-(2,3-dimethylphenyl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
1-benzyl-8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4S)-1-[(6-fluoroquinolin-2-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
1-(1H-indole-5-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
4-(2-methyl-1H-imidazol-1-yl)-1-[3-(2-methylphenoxymethyl)piperidin-1-yl]butan-1-one
2-(2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-6-methyl-2,3-dihydropyridazin-3-one
3-(3-chlorobenzoyl)-1-(furan-3-carbonyl)piperidine
1-[1-(4-methylpentanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
4-(2H-1,3-benzodioxol-5-ylmethyl)-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
(1R,2S,6R,7S)-4-[(4-methoxypyridin-2-yl)methyl]-4-azatricyclo[5.2.2.02,6]undecane
N-methyl-2-(2-oxopiperidin-1-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
1-cyclohexyl-5-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
{4-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-1-methylpiperazin-2-yl}methanol
2-(3-methylbutyl)-8-(morpholine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
9-methoxy-7-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-3-[(2,4,5-trimethylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyrrolidin-1-yl)propan-1-one
methyl (2S,4R)-4-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamido}-1-methylpyrrolidine-2-carboxylate
5-acetyl-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}thiophene-2-carboxamide