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3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
4-(4-butylphenyl)-4H-1,2,4-triazole
1-[5-(methoxymethyl)furan-2-carbonyl]-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
6-[methyl({2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl})amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
5-methyl-4-[(4-methyl-1H-pyrazol-1-yl)methyl]-2-(3-methylthiophen-2-yl)-1,3-oxazole
2-methyl-5-{4-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-cyclopropyl-4-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}pyrrolidin-2-one
3-[(2-fluoro-5-methoxyphenyl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3-phenyl-1,2,4-oxadiazole
2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-methylthiophene-2-carboxamide
4-{1-[6-(4,4-dimethylpiperidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclohexyl-N-(prop-2-yn-1-yl)-1,2-oxazole-5-carboxamide
4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazole
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
(2R,6R)-4-[(3-hydroxy-4-methoxyphenyl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
4,6-dimethoxy-2-[3-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidine
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-methyl-1H-pyrazole-5-carboxamide
2-[3-(dimethylamino)propyl]-9-(quinolin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S,4R)-4-propyl-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanesulfonamide
2-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
1-methyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
(2E)-N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(3-fluorophenyl)prop-2-enamide
(2R)-2-hydroxy-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-2-phenylacetamide
4-methoxy-N-[2-methyl-2-(morpholin-4-yl)propyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
2-[(1S,5R)-3-[4-(1H-imidazol-1-yl)butanoyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
methyl 4-(4-{[(adamantan-1-ylmethyl)(2-hydroxyethyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
5-(4-methyl-1H-pyrazol-1-yl)furan-2-carboxylic acid
3-[2-amino-4-methyl-6-({[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}amino)pyrimidin-5-yl]propanoic acid
1-[2-(4-methoxyphenyl)ethyl]-8-[(3-methoxyphenyl)methyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-6-methyl-3-[3-(piperidin-4-ylmethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-5-chloro-3-ethyl-1-methyl-1H-pyrazole
1-(naphthalen-1-ylmethyl)-N-[(3S)-piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
1-(4-benzylpiperazin-1-yl)-3-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]propan-1-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(dimethyl-1,3-thiazole-5-carbonyl)piperidine-4-carboxylic acid
N-[4-chloro-3-({[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]carbamoyl}amino)phenyl]-2-methoxyacetamide
5-ethoxy-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}furan-2-carboxamide
N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-(1-cyclopentyl-6-oxopiperidine-3-carbonyl)-1-[(3-fluorophenyl)methyl]piperazin-2-one
{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(piperidin-1-yl)ethyl]amine
3-butyl-4-(3-fluoro-4-methoxybenzoyl)-1-methylpiperazin-2-one
1-(4-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-4-oxobutyl)piperidin-2-one
5-methyl-N-[2-(methylsulfanyl)ethyl]-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-(furan-2-ylmethyl)-1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine