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[(2S)-1-{6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}pyrrolidin-2-yl]methanol
8-(2-ethoxypyridine-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-3-carboxamide
5-methoxy-2-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenol
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2,2-diphenylacetamide
4-(4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-2-methylbutan-2-ol
2-{1-[(4-fluorophenyl)methyl]-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
2-amino-6-cyclobutyl-4-[2-(ethylsulfanyl)pyrimidin-5-yl]pyridine-3-carbonitrile
(2S,4R)-N-[2-(2-fluorophenyl)ethyl]-4-{[(2-hydroxyphenyl)methyl]amino}-1-(2-methylpropyl)pyrrolidine-2-carboxamide
1-{1-[3-(furan-3-yl)phenyl]ethyl}pyrrolidine
2-methyl-7-(trimethylpyrimidin-4-yl)-2,7-diazaspiro[4.4]nonane
(2S,4R)-4-amino-N-ethyl-1-[(2-hydroxy-7-methylquinolin-3-yl)methyl]pyrrolidine-2-carboxamide
3-(2-fluorophenyl)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propan-1-one
5-[3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
4-(2,2-dimethyloxane-4-carbonyl)-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(propyl)(pyridin-3-ylmethyl)amine
1-[1-(furan-2-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
methyl 4-({4-[5-(3-methylbutanamido)-1H-pyrazol-1-yl]piperidin-1-yl}methyl)benzoate
1-(4-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-4-oxobutyl)piperidin-2-one
4,4,4-trifluoro-1-(3-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)butan-1-one
(3R,4R)-1-[4-(azepan-1-ylmethyl)benzoyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
4-(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidine-3-carbonyl)morpholine
4-(3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)-1,4-diazepane-1-carbaldehyde
2-{2,7-diazaspiro[4.5]decane-7-carbonyl}-N-(pyridin-2-ylmethyl)aniline
3-(2-methoxyethyl)-5-[(2S)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
1-(4-fluorophenyl)-6,6-dimethyl-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-[(4-methyl-6-{[1-(1,3-thiazol-2-yl)propyl]amino}pyrimidin-2-yl)amino]phenol
N-[(1R)-1-(4-methoxyphenyl)ethyl]-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2-{4-[(2-chloro-6-fluorophenyl)methyl]morpholin-3-yl}acetic acid
4-methyl-1-{2-[4-(3-methylphenoxy)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
4-(4-fluorophenoxy)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
6-chloro-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
4-({1-[(2-hydroxy-6-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
N-[(4-methylphenyl)methyl]-1-(oxolane-3-carbonyl)piperidine-4-carboxamide
methyl 5-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-{3-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-oxopropyl}piperidin-2-one
ethyl 1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-3-(2-methoxyethyl)piperidine-3-carboxylate
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-hydroxypyridine-3-carboxamide
N-{[5-({ethyl[(3R,4R)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]amino}methyl)furan-2-yl]methyl}-N-methylmethanesulfonamide
2-(3,5-dimethoxyphenyl)-N-methylpyridine-4-carboxamide
5-[benzyl(methyl)amino]-2-(1,4-dioxan-2-ylmethyl)-2,3-dihydropyridazin-3-one
3-(5-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
N-cyclopentyl-2,4-difluoro-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzene-1-sulfonamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(1-methoxypropan-2-yl)-5-methyl-1H-pyrazole-4-carboxamide
methyl 5-{[(2,4-dimethoxyphenyl)methyl]amino}-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[5-(ethylcarbamoyl)pyridin-2-yl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-4-carboxamide
2-{[(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)oxy]methyl}pyridine