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4-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]oxane-4-carbonitrile
1-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}-4-(4-fluorophenyl)piperazine
N-(2-{7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]-6-methylpyridine-2-carboxamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
4-phenyl-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperidine-4-carbonitrile
1-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
4-benzyl-1-methyl-3-[1-(pyrimidine-4-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-cyclohexyl-2-[(3-methoxyphenyl)methyl]morpholine
5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-N-(pyrrolidin-3-yl)pyridin-2-amine
1-[2-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-oxoethyl]-1,2-dihydropyrimidin-2-one
3-benzyl-7-(2,6-dimethylhept-5-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-{1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]piperidin-4-yl}methanesulfonamide
5-chloro-4,6-dimethyl-2-oxo-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}cyclohexanecarboxamide
N-(3-methoxyphenyl)-3-{1-[3-(1H-pyrazol-4-yl)propanoyl]piperidin-4-yl}propanamide
methyl 1-(2-methylpropyl)-3-(pyridine-3-amido)-5-[(thiophen-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]-4-ethylpiperazine-2,3-dione
4-(pyridin-4-yl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}pyrimidin-2-amine
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 4-[1-(quinoxaline-6-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
6-{2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-2-carbonitrile
3-(hydroxymethyl)-N-methyl-N-[(4-phenoxyphenyl)methyl]benzamide
2-{4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazin-1-yl}-1-(pyrrolidin-1-yl)ethan-1-one
1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
1,3-dimethyl-2,6-dioxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-{2-methoxy-5-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]phenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
1-[1-ethyl-5-(2,3,6-trifluorobenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
2-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]benzonitrile
N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-(piperidin-1-yl)benzamide
N-[1-(4-fluorophenyl)-5-oxopyrrolidin-3-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
ethyl 1-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}piperidine-4-carboxylate
8-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
N-(cyclopropylmethyl)-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
2-amino-6-{4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
5-(2-fluorophenyl)-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}-1,2,4-triazin-3-amine
1-({1-[6-(pyrimidin-5-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-5-(4-fluorophenyl)-4-phenyl-1H-imidazole
1-(2-chloro-4,5-difluorobenzoyl)-3-(2-methoxyphenoxy)azetidine
1-(cyclohexylmethyl)-6-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]piperidine-3-carboxamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
5-(1-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}pyrrolidin-2-yl)-N,N-dimethylthiophene-2-carboxamide
(4-{[2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl}-1,4-oxazepan-6-yl)methanol
4-{[ethyl(oxan-4-yl)amino]methyl}-1H-pyrazole-3-carboxylic acid
(1R,5R)-3-(pyrazin-2-yl)-6-[(2,3,4-trifluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-(2-fluorophenyl)-3-phenyl-N-[2-(propane-2-sulfonyl)ethyl]propanamide
N-(3-{[(2,2-dimethyloxan-4-yl)(ethyl)carbamoyl]methoxy}phenyl)propanamide
2-(3-methyl-1H-pyrazol-1-yl)-1-{4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one