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5-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]-2-(methylsulfanyl)pyrimidine
3-(3,5-difluoro-2-methoxyphenyl)pyrazolo[1,5-a]pyrimidine
N-[1-(3,3-dimethylbutyl)azepan-4-yl]-1,3,5-trimethyl-1H-pyrazole-4-sulfonamide
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]pyrimidin-2-amine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(2-{[4-(propan-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenoxy)ethan-1-ol
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-methyl-3-phenylpiperidine
1-{6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-3-yl}ethan-1-one
9-[2-(propan-2-yloxy)acetyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
9-[(4-methoxy-2-methylphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-{2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamido}butanoate
3-[({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)methyl]-1λ6-thiolane-1,1-dione
ethyl 1-cyclobutanecarbonyl-4-[(3-fluorophenyl)methyl]piperidine-4-carboxylate
2-chloro-4-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}-6-methoxyphenol
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-(pyrrolidine-1-carbonyl)piperidin-4-amine
5-[(4-hydroxyphenyl)methyl]-N-[(4-methoxyphenyl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-benzyl-3-ethyl-1-(2-hydroxy-4-methoxybenzoyl)-1,4-diazepan-5-one
N-ethyl-2-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-N-methylacetamide
2-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
N-(2-ethoxyphenyl)-N'-[2-(pyridin-4-ylformamido)ethyl]propanediamide
6-(aminomethyl)-N,2-dimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine
6-chloro-4-(4-methoxypiperidin-1-yl)-2-[(2-methyl-4-phenylpiperazin-1-yl)methyl]quinazoline
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)acetamide
2-(4-fluorophenyl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]imidazo[1,2-a]pyridine-6-carboxamide
5-[6-(trifluoromethyl)pyridin-3-yl]pyridin-3-amine
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2-methoxyacetamide
1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
(4aS,7aR)-1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(7-fluoro-4-methylquinolin-2-yl)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-phenylpyrrolidin-3-ol
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N,1-dimethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyrrolidine-3-carboxamide
8-{2-[4-(dimethylamino)phenyl]acetyl}-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[1-(5-acetylthiophene-2-carbonyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
(5R)-5-[6-methyl-5-(5-phenyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl]pyrrolidin-2-one
N,N-diethyl-1-{1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
4-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydroisoquinolin-1-one
1-(1-ethyl-1H-pyrazole-3-carbonyl)-3,3-diphenylpiperidine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(2,2-dimethyloxan-4-yl)-N-ethyl-1H-pyrazole-3-carboxamide
4-(4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-1-phenyl-1H-pyrazol-3-yl)pyridine
N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
[(3-{[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](furan-3-ylmethyl)methylamine
1-cyclopentyl-4-[4-(piperidin-3-ylmethyl)benzoyl]-1,4-diazepane
N-[(2R,3R)-1'-[(5-chloro-2-hydroxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(pyridin-4-ylsulfanyl)acetamide
N-[2-(1H-indol-3-yl)ethyl]-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-{[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]sulfamoyl}-N-(pyridin-3-yl)benzamide
methyl (2S,4R)-1-({3-[(acetyloxy)methyl]-4-ethoxyphenyl}methyl)-4-hydroxypyrrolidine-2-carboxylate
(1S)-1-[1-(3-methylphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
(1S,5R)-N-(2-ethoxyphenyl)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide