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N-(2-fluorophenyl)-3-[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]propanamide
4-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-N,N-dimethylmorpholine-2-carboxamide
1-[(2-chlorophenyl)methyl]-N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
11-[butyl(methyl)amino]-4-[2-(3-methoxyphenyl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-[(3R,4S)-1-[(6-methylquinolin-5-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-(2-fluorophenyl)-N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-4-carboxamide
2-(2-methoxyethyl)-9-(1-methyl-1H-indole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S,5S)-1-(3-methyl-1H-pyrazole-5-carbonyl)-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
1-(2,4-dimethylphenoxy)-3-[(2-methyloxolan-3-yl)amino]propan-2-ol
(2S,4S)-N-cyclopropyl-1-[(2,3-dimethoxyphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carboxamide
N-methyl-1-propyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(6-methylpyridine-3-carbonyl)piperidine-4-carboxylic acid
4-{2-[1-ethyl-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}-1λ6-thiomorpholine-1,1-dione
ethyl 4-(3-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propoxy)benzoate
5-butyl-1'-(3-ethyl-1,2-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[2-(oxolan-2-ylmethoxy)phenyl]acetamide
2-{4-[1-(thiophene-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
3,5,7-trimethyl-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
4-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2,3-dihydro-1H-imidazol-2-one
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[(3-methylquinoxalin-2-yl)methyl]pyrrolidin-3-yl]methanol
3-[2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1,2-dihydroquinolin-2-one
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-2-(propan-2-yloxy)propanamide
[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
(3aR,6aR)-2-methanesulfonyl-5-{6-methylthieno[2,3-d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{2-[2-(2-methoxyethyl)morpholin-4-yl]-2-oxoethyl}-1,2-dihydroisoquinolin-1-one
2-(5-methoxy-1,3-benzoxazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-5-[(methylsulfanyl)methyl]-N-(quinolin-5-ylmethyl)furan-2-carboxamide
N-[(7-{[2-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-2-phenylacetamide
1-{[1-(4-methoxyphenyl)-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,4-diazepane
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-(3-methoxyphenyl)-N-methyl-1,2,4-triazin-3-amine
4-(1-methyl-1H-imidazol-2-yl)-1-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperidine
methyl 3-(3-chlorobenzamido)-6-(thiomorpholin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
2-{4-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]phenyl}acetic acid
3-[({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)methyl]phenol
(3S,4S)-1-{2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(dimethylamino)pyrrolidin-3-ol
2-(3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)-6-methylpyridine-3-carbonitrile
2-(azepan-1-yl)-2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}acetic acid
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-(4-methoxyphenyl)-1,2,4-triazin-3-amine
2-{4-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-6-hydroxy-1,4-diazepan-1-yl}acetic acid
methyl 3-({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)-5-methoxybenzoate
8-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-[(2-aminopyridin-3-yl)methyl]-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)benzamide
(3R,4S)-4-cyclopropyl-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)pyrrolidin-3-amine
7-(pyridine-3-carbonyl)-N-[2-(pyrrolidin-1-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[3-(4-fluorophenoxymethyl)-5-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amine
dimethyl[({1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}methyl)sulfamoyl]amine