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4-(2,5-dimethoxyphenyl)-2-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]phenol
2-(2H-1,2,3-benzotriazol-2-yl)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}acetamide
3-(4-methoxyphenyl)-N-{[8-(propan-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
5-[1-(3-methylbenzoyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
N-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-N-[(3-methylthiophen-2-yl)methyl]cyclopentanamine
N,1,3-trimethyl-N-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-2-phenylethyl]-1H-pyrazole-5-carboxamide
N-(2-phenoxyethyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydroquinazolin-4-one
[1-({1-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
5-methyl-5-{1-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]piperidin-4-yl}-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
2-{1-[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-triazin-3-yl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
2-(dimethylamino)-N-[5-({[3-(1H-imidazol-2-yl)propyl]carbamoyl}amino)-2-methylphenyl]acetamide
1-ethyl-5-(1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-4-phenyl-1H-imidazol-5-yl)-1H-1,2,4-triazole
1-cyclopentyl-N-[2-(4-methoxyphenyl)ethyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-({4-methyl-5-[1-(pyridine-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-{1-cyclopentyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenol
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
6-methyl-5-{[3-(2-methylpropyl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(methylamino)-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]pyridine-4-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(1,2-oxazinan-2-yl)propanamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(6-fluoropyridin-3-yl)-1-(3-methoxypropyl)-1-[(4-methylphenyl)methyl]urea
(1R,5R)-6-(cyclobutylmethyl)-3-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonane
(2R,3S,6R)-5-[1-(methoxymethyl)cyclobutanecarbonyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[1-benzyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]-1-methylpiperidin-4-ol
2-[1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazol-5-yl]-1H-1,3-benzodiazole
7-[(3-chloro-4-fluorophenyl)methyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-methyl-5-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyrimidin-2-amine
3-methyl-2-(3-methylphenoxy)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]butan-1-one
1-[3-(2-methylpyrimidin-4-yl)phenyl]-N-[2-(thiophen-2-yl)ethyl]piperidin-4-amine
3-(4-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenyl)prop-2-yn-1-ol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(1S,3R)-3-amino-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]cyclopentane-1-carboxamide
N-methyl-2-[(prop-2-en-1-yl)amino]-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
N-{1-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-(pyrrolidin-1-yl)piperidine
(2S,4R)-N-methyl-4-(4-{[N-methyl-1-(3-methylthiophen-2-yl)formamido]methyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]amine
5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-oxazole-3-carboxamide
(2-ethoxy-5-{[2-(2-methoxyethyl)piperidin-1-yl]methyl}phenyl)methanol
2-{[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]methyl}-6-methoxyphenol
N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-amine
3-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-1-{4-[(trifluoromethyl)sulfanyl]phenyl}urea
2-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(dimethylamino)-1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-(4-methylphenyl)ethan-1-one
4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
2-(2-amino-2-methylpropanoyl)-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide