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2-(4-methoxyphenoxymethyl)-4-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1,3-oxazole
7-cyclopentyl-2-[2-(methylsulfanyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
1-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]urea
{[(3R,4S)-4-cyclopropyl-1-[(3-methylpyrazin-2-yl)methyl]pyrrolidin-3-yl]sulfamoyl}dimethylamine
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(quinolin-5-yl)pyridine-3-carbonitrile
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine
8-(2,3-dihydro-1H-inden-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
(4aR,7aS)-1-(2-{[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-(2-methyl-6-propylpyrimidin-4-yl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]piperidin-4-amine
5-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
2-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-4-(pyridin-3-yl)pyrimidine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
2-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}-3-methoxyphenol
1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
2-methoxy-1-{4-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
5-(4-acetylphenoxymethyl)-N-(2-hydroxy-2-phenylethyl)-N-methyl-1,2-oxazole-3-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]pyrimidin-4-amine
2-({1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
N-ethyl-1-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}pyrrolidine-3-carboxamide
1-ethyl-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-cyclopropyl-N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-2-methylpropanamide
2-{4-[(3-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}acetamide
ethyl 3-(3-phenylpropyl)-1-(thiophene-3-carbonyl)piperidine-3-carboxylate
6-(hydroxymethyl)-N-(isoquinolin-5-ylmethyl)-N-methylpyridine-2-carboxamide
2-amino-4-ethyl-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-1,3-thiazole-5-carboxamide
N-{2-[4-({[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}methanesulfonamide
2-(4-cyclohexylpiperazine-1-carbonyl)-5-fluoro-1,3-dimethyl-1H-indole
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(3-fluorophenyl)-N-methyl-N-(oxan-2-ylmethyl)-1,3-benzoxazole-5-carboxamide
3-(3-chlorophenyl)-N-[(5-methylpyrazin-2-yl)methyl]-3-phenylpropanamide
2,6,8-trimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)quinoline-4-carboxamide
(3aR,5R,6S,7aS)-N-[2-(4-fluorophenoxy)phenyl]-5,6-dihydroxy-octahydro-1H-isoindole-2-carboxamide
dimethyl(3-{2-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}morpholine-2-carboxylic acid
2-(5-acetylthiophen-3-yl)-N-{[4-(trifluoromethoxy)phenyl]methyl}acetamide
(2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-1,3-thiazol-4-yl)methanol
N3-[2-(3-fluorophenyl)ethyl]-N5-[(4-fluorophenyl)methyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(cyclopentylmethyl)-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
7-methyl-3-[(4-methyl-1,4-diazepan-1-yl)methyl]-2-(thiophen-2-yl)quinoline
3-fluoro-5-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
7-(cyclopropylmethyl)-2-(2-methyl-1-benzofuran-5-carbonyl)-2,7-diazaspiro[4.5]decane
4-(2-methylphenoxy)-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxylic acid
1-{[3-(difluoromethoxy)phenyl]methyl}-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
(1R,5R)-6-[(5-ethylpyridin-2-yl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane