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N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
2-(2-methoxyethoxy)-1-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
1-(4-fluorophenyl)-4-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]piperazine
3-[1-(2-acetylbenzoyl)piperidin-3-yl]-N-(3,5-dimethoxyphenyl)propanamide
2-(dimethylamino)-4-methyl-N-[2-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
6-(3-oxo-3-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propyl)-2,3,4,5-tetrahydropyridazin-3-one
2-cyclopropyl-8-(3-hydroxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-chloro-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]pyridine-4-carboxamide
1-(oxane-2-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
2-methyl-4-phenyl-3-[3-(pyrrolidin-1-yl)piperidine-1-carbonyl]pyridine
2-(dimethylamino)-N-methyl-2-(2-methylphenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
N3-cyclooctyl-N5-(2-methylpropyl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(4aR,7aS)-1-(3-methylbutanoyl)-4-(5-methylpyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(pyridin-3-ylmethyl)({[6-(trifluoromethyl)pyridin-3-yl]methyl})amino]butan-1-ol
N-{4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}ethane-1-sulfonamide
4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}morpholine
1-(2-methoxyethyl)-8-methyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
ethyl 1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,2,5-thiadiazole-3-carboxamide
5-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}pyrimidine
5-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,3-dimethyl-1H-pyrazole
1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(furan-2-carbonyl)piperazine
2-[6-(methoxymethyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
1-{2-[1-butyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]phenyl}-1,3-diazinane-2,4-dione
1-{2-oxo-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
4-(4-methoxyphenoxy)-1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperidine
(2S,4R)-4-amino-1-{[2,5-dimethyl-1-(4-methylpyridin-2-yl)-1H-pyrrol-3-yl]methyl}-N-methylpyrrolidine-2-carboxamide
(2S,4R)-1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-4-amino-N,N-diethylpyrrolidine-2-carboxamide
N-(3-hydroxypropyl)-1-methyl-2-oxo-N-(pyridin-4-ylmethyl)-1,2-dihydroquinoline-3-carboxamide
(3aR,6aR)-2-[(4-chlorophenyl)methanesulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[1-({2-[4-(1H-imidazol-1-yl)butoxy]phenyl}methyl)pyrrolidin-2-yl]pyridine
2-[(dimethylcarbamoyl)amino]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
ethyl 4-(5,7-dimethoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-1H-pyrazole-3-carboxylate
(3S,4R)-4-(hydroxymethyl)-1-(1H-indol-5-ylmethyl)piperidin-3-ol
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-(1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
5-[2-(3-methoxypropyl)piperidine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
N-[(2-methylphenyl)(pyridin-4-yl)methyl]-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)-1-azabicyclo[2.2.2]octan-3-amine
N-[(4-methyl-1,4-oxazepan-6-yl)methyl]quinoxalin-2-amine
[3-(cyclopropylmethyl)-1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-3-yl]methanol
(1H-imidazol-2-ylmethyl)[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
8-(oxolan-3-yl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 3-[(3S,4R)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
6-[3-(dimethylamino)benzoyl]-N-[(6-methylpyridin-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-methyl-4-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}imidazolidin-2-one
2-[1-(3-cyclohexyl-1H-pyrazol-4-yl)-N-methylformamido]acetic acid
(4aR,7aS)-1-butyl-4-[(3,5-dimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione