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5-(4-methanesulfonylphenyl)-1-propyl-1H-1,2,4-triazole
2-(cyclopent-1-ene-1-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
4-(5-methylpyridin-2-yl)-1-(pyrimidin-2-yl)piperidin-4-ol
8-(5-chloro-2-methoxybenzoyl)-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
3-methyl-3-phenyl-1-(1,2-thiazole-5-carbonyl)piperidine
{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(4-methoxyphenyl)ethyl]methylamine
N,2-dimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]imidazo[1,2-a]pyrimidine-3-carboxamide
N-(1-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
(2S,4R)-4-amino-1-(3-cyanobenzenesulfonyl)-N,N-diethylpyrrolidine-2-carboxamide
5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,3-benzodiazole-7-carboxamide
N-ethyl-2-[4-(2-oxoimidazolidin-1-yl)phenyl]-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
3-{[(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)amino]methyl}-1λ6-thiolane-1,1-dione
2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-[(pyridin-2-ylmethyl)amino]benzamide
methyl 2-(3-oxo-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazin-2-yl)acetate
2-[1-methyl-10-oxo-4-(piperidine-1-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-(3-hydroxypiperidin-1-yl)ethan-1-one
8-(3,5-difluoropyridine-2-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(1-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}piperidin-3-yl)methanol
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-3-amine
1-(2-chloroprop-2-en-1-yl)-3-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
2-(3-methoxypropyl)-8-[(4-methyl-1H-imidazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
1-{2-[3-(3-methylphenoxy)azetidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl})amine
methyl 1-({2-[2-hydroxy-3-(4-methylpiperazin-1-yl)propoxy]-4-methoxyphenyl}methyl)piperidine-4-carboxylate
N-(1,3-benzoxazol-2-ylmethyl)-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
(3aR,7aS)-5-methyl-2-(5-methylpyrazine-2-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(4aR,8aR)-2-(1H-imidazol-4-ylmethyl)-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
{[7-chloro-2-(2-phenylethoxy)quinolin-3-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl]amine
3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-6-(thiophene-2-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-[1-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1H-imidazol-2-yl]benzonitrile
1-methyl-3-(thiomorpholine-4-carbonyl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{3-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-3-oxopropyl}methanesulfonamide
N-[(3R,4S)-1-(5-cyanopyridin-2-yl)-4-cyclopropylpyrrolidin-3-yl]-4-acetamidobutanamide
N-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-N-methylcyclohexanamine
N-(1-{4-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]phenyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
1-[(4-fluorophenyl)methyl]-N-[2-(furan-2-yl)ethyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
4-{[(1-carbamoylpiperidin-3-yl)formamido]methyl}benzoic acid
3-methyl-7-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-({8-[(2-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)isoquinoline-3-carboxamide
3-methyl-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(pyridin-2-ylmethyl)piperazine
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
4-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
(2S,4R)-N-[3-(benzyloxy)phenyl]-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carboxamide