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N-(1-{[(2,3-dihydro-1H-inden-2-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-3-(2-methoxyphenyl)propanamide
N-{[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
4-[(3-{2-[1-(furan-2-carbonyl)piperidin-2-yl]ethoxy}-4-methoxyphenyl)methyl]morpholine
N5-(2-methoxyethyl)-N3-methyl-1-(3-methylbutyl)-N3-[2-(4-methylphenoxy)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
{[6-(4-ethylpiperazin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}[2-(3-fluorophenyl)ethyl]amine
N-[1-(2,4-dimethoxyphenyl)ethyl]-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]pyridin-2-amine
(2S)-N-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
5-{1-[2-(1H-imidazol-2-yl)benzoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
methyl 6-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}-3-cyclopropaneamidothieno[2,3-b]pyridine-2-carboxylate
1-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-(oxolan-3-yl)-1H-1,2,3-triazole
5-(azocane-1-carbonyl)-1-benzyl-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
(4S)-3-{2-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-2-oxoethyl}-4-phenyl-1,3-oxazolidin-2-one
4-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)benzamide
2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]acetamide
2-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-3-ol
2-(dimethylamino)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
3-{4-[1-(furan-3-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}prop-2-yn-1-ol
2-amino-4-(oxolan-3-yl)-6-[4-(piperidin-1-yl)phenyl]pyridine-3-carbonitrile
2-[1-({2-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)piperidin-3-yl]propan-2-ol
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
methyl 3-(2-chlorobenzenesulfonamido)-5-{[(3-methylphenyl)formamido]methyl}benzoate
3-[1-(4-amino-5-methylpyrimidin-2-yl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(azepan-1-yl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
6-{4-[(4-methylphenyl)sulfanyl]piperidine-1-carbonyl}piperazin-2-one
6-(3-phenoxypropanoyl)-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
5-ethoxy-2-methyl-N-[(1-methylpiperidin-3-yl)methyl]-1-benzofuran-3-carboxamide
3-fluoro-N-[1-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
(3R,4S)-4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(ethyl)amino)oxolan-3-ol
1-({[2-fluoro-5-(trifluoromethyl)phenyl]carbamoyl}amino)-N-methylcyclohexane-1-carboxamide
ethyl 4-[(2-chlorophenyl)methyl]-1-[(4-acetamidophenyl)methyl]piperidine-4-carboxylate
6-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
2-{4-[(2,5-difluorophenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
3,5-difluoro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-methoxybenzamide
1-(furan-2-ylmethyl)-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]piperidine-4-carboxamide
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)[2-(1H-imidazol-1-yl)ethyl]methylamine
4-[(4-fluorophenyl)methyl]-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3-(propan-2-yl)-1,4-diazepan-5-one
9-[(2S,3R)-2-amino-3-hydroxybutanoyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
[5-(2H-1,3-benzodioxol-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
3-cyclopropyl-1-(6-hydroxy-4-{thieno[3,2-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)propan-1-one
N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-{furo[3,2-c]pyridin-4-yl}piperidine
2-phenyl-1-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl)ethan-1-one
1-(2-{[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
9-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(2-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)benzene-1-sulfonamide
8-chloro-2-{[(thiolan-3-yl)amino]methyl}quinolin-4-ol