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6-(cyclohex-3-en-1-ylmethyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-(1H-indol-1-yl)ethyl]benzamide
[(4-ethynylphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
1-[(2-chlorophenyl)methyl]-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-{3-[1-(dimethylamino)ethyl]phenyl}-N,N-dimethyl-1H-1,2,4-triazol-5-amine
methyl (2S)-3-methyl-2-[(1-methyl-1H-pyrazol-5-yl)formamido]butanoate
1-[(1-hydroxycyclohexyl)methyl]-3-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]urea
4-{[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]methyl}-2,6-dimethoxyphenol
6-[4-(4-chlorophenoxy)piperidin-1-yl]pyrimidine-2,4-diamine
5-(4-chloro-2-methoxyphenoxymethyl)-N-(1-hydroxybutan-2-yl)-1,2-oxazole-3-carboxamide
3-{2-[4-(3-chloro-4-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
2-(methylsulfanyl)-5-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}pyrimidine
2-(1-{imidazo[1,2-a]pyridine-3-carbonyl}piperidin-3-yl)-4-methyl-1H-1,3-benzodiazole
2-{1-[(4-methylphenyl)methyl]-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
1-(thiophene-2-carbonyl)-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
1-{7-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,2,3,6-tetrahydropyridine
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
3-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
(3S,4S)-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
1-[1'-(5-ethyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
6-methyl-5-{2-oxo-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1,4-oxazepan-6-yl]methanol
ethyl 4-{6-[(5-acetamidothiophen-2-yl)methyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
5-methyl-N-[phenyl(pyridin-4-yl)methyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-(5-methylfuran-2-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-pyrazole-5-carboxamide
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]cyclopropanecarboxamide
6-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N4-(furan-3-ylmethyl)-N2,N2,N4-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-3-[(2,4,5-trimethylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
6-oxo-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-ethyl-5-[4-(2-methylphenoxy)piperidine-1-carbonyl]pyrimidin-2-amine
(3aS,6aS)-2-(2-methoxyethyl)-5-(2-phenylethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(azepan-1-yl)-2-phenylethyl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(4-methylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
7-chloro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-methyl-1H-indole-2-carboxamide
4-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}benzoic acid
1-({5-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]furan-2-yl}methyl)-1H-imidazole
3-[2-(azocan-1-yl)-2-oxoethyl]-3-(2-chlorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
4-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-ethyl-9-[(5-ethylthiophen-2-yl)sulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(4-methoxyphenyl)-N-[2-(oxan-3-yl)ethyl]-1H-pyrazole-5-carboxamide
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-(4-phenoxybenzoyl)piperidine
methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)[2-(oxan-4-yl)ethyl]amine
{1-[3-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)propyl]piperidin-2-yl}methanol