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3-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-1,4-dihydropyridin-4-one
ethyl 2-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]amino}acetate
(3S,5R)-1-benzyl-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
1-({5-[(3,5-dimethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
2-(1-methyl-1H-indol-3-yl)-N-propyl-N-(pyridin-3-ylmethyl)acetamide
(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl](pyridin-2-ylmethyl)amine
4-(3-{3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}phenyl)morpholine
2-fluoro-N-methyl-5-[({[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}carbamoyl)amino]benzamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
5-ethyl-2-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrimidin-4-amine
6-methyl-4-oxo-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-4H-pyran-2-carboxamide
2-(2-{[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
N-(1,5-dimethyl-1H-pyrazol-4-yl)-4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carboxamide
(3aR,6aR)-2-(2,5-difluorobenzoyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-7-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-N-(propan-2-yl)-1,4-dihydro-1,8-naphthyridine-3-carboxamide
N-(2,2-dimethyloxan-4-yl)-N-ethyl-3,5-dimethyl-1H-indole-2-carboxamide
1-(3-chloro-4-methoxyphenyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
2-methyl-5-[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
N-[2-(2-phenoxyphenyl)ethyl]oxolane-3-carboxamide
2-(4-{[(3R)-3-aminopyrrolidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
4-{1-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-imidazol-2-yl}pyridine
4-methyl-2-(4-methylpiperazin-1-yl)-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)pyrimidine
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[3-chloro-2-(4-ethylpiperazin-1-yl)phenyl]acetamide
ethyl 4-[(3-fluorophenyl)methyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-4-carboxylate
N-(cyclobutylmethyl)-7-acetamido-1-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]-N5-(oxolan-2-ylmethyl)piperidine-3,5-dicarboxamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-indole-6-carboxamide
N-methyl-5-oxo-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-[(2-methoxyethyl)sulfanyl]-5-(3-methoxyphenyl)-4-[1-(pyrazine-2-carbonyl)piperidin-3-yl]pyrimidine
2-(3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenyl)-3,4,5,6,7,8-hexahydroquinazolin-4-one
N-(4-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}-3-methylphenyl)acetamide
N-methyl-N-(2-phenyl-1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}ethyl)thiophene-2-carboxamide
1-(2-chlorophenyl)-3-{[1-(ethoxymethyl)cyclobutyl]methyl}urea
N-[(2,4,5-trifluorophenyl)methyl]oxolane-3-carboxamide
N-ethyl-N-[1-(4-methoxyphenyl)propyl]pyridine-4-carboxamide
5-(2-fluorophenyl)-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
4-{1-benzyl-5-[1-(propan-2-yl)piperidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
3,5-dichloro-N-methyl-4-(prop-2-en-1-yloxy)-N-(prop-2-yn-1-yl)benzamide
2-phenoxy-N-(2-{7-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
2-{[2-(trifluoromethyl)pyrrolidin-1-yl]methyl}pyridine-3-carboxylic acid
5-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-3-(2,3-dihydro-1H-inden-2-yl)-5-methylimidazolidine-2,4-dione
8-methyl-N-(2,4,4-trimethylpentan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-ethyl-3-methyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}furan-2-carboxamide
1-(cyclopropanesulfonyl)-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
(furan-2-ylmethyl)(methyl){[3-(thiophen-3-yl)-1H-pyrazol-5-yl]methyl}amine
N-[(3S,5S)-5-(azepane-1-carbonyl)-1-methylpyrrolidin-3-yl]-3-methoxypropanamide
N-[(3-hydroxyphenyl)methyl]-3-methoxy-N,2,2-trimethylpropanamide
1-ethyl-N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1H-pyrazole-4-carboxamide
8-(isoquinoline-5-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one