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2-{4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
{4-[(2-chlorophenyl)methyl]-1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperidin-4-yl}methanol
1-[(6-ethylpyrimidin-4-yl)amino]-3-(piperidin-1-yl)propan-2-ol
1-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-3-(1H-imidazol-2-yl)piperidine
benzyl(2-phenylethyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
5-{[(4-fluorophenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(2,6-dimethylphenyl)-2-[(2-methoxyethyl)(methyl)amino]acetic acid
4-{2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-5-fluoropyrimidin-4-yl}morpholine
N-{[2-(3-chlorophenyl)-7-methylquinolin-3-yl]methyl}-N-(3-methoxypropyl)furan-2-carboxamide
(3S,4R)-1-(3-fluoro-4-methoxybenzoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-methyl-3-phenyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
8-methyl-2-propyl-3-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2,8-diazaspiro[4.5]decane
dimethyl[2-({[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}(thiophen-3-ylmethyl)amino)ethyl]amine
2-methoxy-6-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}phenol
4-[2-(3-chlorophenyl)-2-hydroxyacetyl]-1-cyclopentylpiperazin-2-one
(4aS,7aR)-4-butyl-6,6-dioxo-N-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(3S,4R)-1-[(5-acetylthiophen-3-yl)methyl]-4-(2H-1,3-benzodioxol-5-yl)pyrrolidine-3-carboxylic acid
5-(1-cyclopentylpyrrolidin-2-yl)-N-[2-(1H-imidazol-1-yl)ethyl]thiophene-2-carboxamide
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[3-(pyridin-3-yl)azetidin-1-yl]butan-1-one
4-[(furan-2-ylmethyl)amino]-5-methyl-N-[2-(pyridin-4-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-(9-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)acetamide
5-phenyl-N-[4-(4-{[3-(pyridin-3-yl)propyl]amino}piperidin-1-yl)phenyl]pentanamide
1-ethyl-6-methyl-2-oxo-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(2-methyl-1H-indol-3-yl)ethan-1-one
3-[5-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]phenol
methyl 3-acetamido-5-[(oxan-4-yl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl](methyl)(3,3,3-trifluoropropyl)amine
(2S,4S)-4-acetamido-N-ethyl-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
[(4-methanesulfonylphenyl)methyl](methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-methyl-5-[2-(2-methylphenyl)acetyl]-N-[3-(morpholin-4-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(5-{1-[(3,5-dichloropyridin-4-yl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
2-{[3-(difluoromethoxy)phenyl]methyl}-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(1-hydroxy-2-methylpropan-2-yl)amino]methyl}piperidin-2-one
4-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-(2,4-dichlorophenoxy)-1-(2-methyl-1,4-oxazepan-4-yl)ethan-1-one
5-butyl-4-(dimethyl-1,2-oxazole-4-carbonyl)-1-(3-methylphenyl)piperazin-2-one
(4aR,8aR)-2-(2,5-dimethylfuran-3-carbonyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-[1-(3,5-difluorophenyl)cyclopropyl]spiro[2.2]pentane-1-carboxamide
N-{2-[2-(piperidin-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-4-(trifluoromethyl)benzamide
5-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-methyl-2-(pyridin-3-yl)pyrimidine
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-4-methyl-N-[(3S)-2-oxoazepan-3-yl]benzamide
4-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-2-yl)-3,5-dimethyl-1,2-oxazole
1-[4-(1H-imidazol-1-yl)butanoyl]-4-phenoxypiperidine-4-carboxylic acid
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}propanamide
methyl 4-({2-[(3-oxo-4-phenylpiperazin-1-yl)methyl]quinazolin-4-yl}amino)butanoate
2-{[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]amino}-N-(3-fluoro-2-methylphenyl)acetamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
N-cyclopropyl-6-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-(2,3-dimethylpyridin-4-yl)-3-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)benzamide