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N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(2H-1,2,3,4-tetrazol-2-yl)acetamide
4-(1H-imidazol-1-yl)-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
(2S,4R)-4-amino-1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-methylpyrrolidine-2-carboxamide
N,2-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-methoxy-2-phenyl-N-{1-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
3-(2-fluorophenyl)-5-(thiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-(2,5-dimethoxyphenyl)-1-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}ethan-1-one
3-amino-N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}butanamide
8-(2,3-dihydro-1H-inden-2-yl)-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(6-methoxypyridin-2-yl)-2-(morpholin-4-ylmethyl)phenol
3-[4-(3-hydroxypiperidin-1-yl)piperidine-1-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
4-[(3-methylphenyl)sulfanyl]-1-(1H-1,2,3-triazole-5-carbonyl)piperidine
7-fluoro-N,3-dimethyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-benzofuran-2-carboxamide
4-{1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrimidin-2-amine
4-{4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
{2-[(1H-imidazol-2-ylmethyl)[(2-methylphenyl)methyl]amino]ethyl}dimethylamine
3-{1-[(4-acetamidophenyl)methyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
(4aS,7aR)-1-[(3-chloro-2,4-difluorophenyl)methyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methoxy-N-(2-methoxyethyl)-2-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-(2-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}quinolin-6-yl)acetamide
N-(2-methoxyethyl)-5-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(1S,5R)-3-(4-hydroxybenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-({4-[(3,5-dimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
(4aS,8aR)-1-(2-aminoethyl)-6-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
5-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}pyridin-2-amine
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidine
5-(2,5-dimethylphenoxymethyl)-N-[2-(1H-indol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[2-(3-methylthiophen-2-yl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
2-(2,4,6-trimethoxyphenyl)-1H-1,3-benzodiazole-6-carboxylic acid
3-(2H-1,3-benzodioxole-5-carbonyl)-1-(oxane-4-carbonyl)piperidine
2-methyl-5-[2-(1H-pyrazol-3-yl)phenyl]-1,3,4-thiadiazole
1-[3-(1H-pyrazol-1-yl)benzoyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-benzyl-1-{2-[2-(2-methoxyphenyl)acetamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
8-(1-methoxypropan-2-yl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-[2-(dimethylamino)ethyl]-2-methoxybenzamide
methyl 2-{3-[(3,4-dimethylphenyl)amino]piperidine-1-carbonyl}benzoate
4-methoxy-N-methyl-N-(oxan-2-ylmethyl)-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[(2-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
6-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]quinoxaline
2-(2-methoxyethyl)-N-(2-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
({5-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]furan-2-yl}methyl)dimethylamine
1-(4-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}piperidin-1-yl)ethan-1-one
4-chloro-5-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide