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4-{5-[({1-[(3-methoxyphenyl)methyl]piperidin-3-yl}amino)methyl]thiophen-2-yl}-2-methylbut-3-yn-2-ol
2-(4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepan-1-yl)-1,3-benzothiazole
4-{3-[(dimethylamino)methyl]phenyl}-7-(2-oxo-1,3-oxazolidin-3-yl)-1,2,3,4-tetrahydroquinolin-2-one
2-(3-fluorophenyl)-N-(1-{4-[4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
6-propyl-2-(3-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-(3-butanamidophenyl)-3-(hydroxymethyl)-4-methylpiperazine-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6-methylquinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
7-[(2,3-difluorophenyl)methyl]-2-(5-methylthiophene-2-carbonyl)-2,7-diazaspiro[4.5]decane
4,6-dihydroxy-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]pyridine-3-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2-(pyridin-4-ylsulfanyl)acetamide
2-butyl-8-[2-(2-hydroxyethoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl (2S)-2-(3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)-2-phenylacetate
N-(oxolan-3-yl)-4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)propanamide
2-[(2-chloro-6-fluorophenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5-{3-[2-(4-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
1-{1-[2-(4-hydroxyphenyl)acetyl]piperidin-3-yl}-3-phenylpropan-1-one
2-cyclopentyl-9-(3-hydroxy-2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-methoxypyridine-3-carbonitrile
9-[3-(dimethylamino)-2,2-dimethylpropyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
8-methoxy-2-{[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}quinoline
(furan-2-ylmethyl)[(6-methoxypyridin-3-yl)methyl](thiophen-3-ylmethyl)amine
5-(4-acetyl-1,4-diazepane-1-carbonyl)-1-[(4-chlorophenyl)methyl]piperidin-2-one
ethyl 1-[2-(3-methylbenzamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carbonyl]piperidine-3-carboxylate
(1S,5R)-6-(cyclopropylmethyl)-3-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(4R)-N,3-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,3-thiazolidine-4-carboxamide
2-(4-chlorophenyl)-N-methyl-N-(pyrazin-2-ylmethyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[2-(morpholin-4-yl)ethyl]-5-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)piperidin-2-one
(3S,4S)-4-methyl-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidine-3,4-diol
2-ethyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)butanamide
1-(4-fluorophenyl)-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)cyclopropane-1-carboxamide
2-methyl-8-{[5-(1H-1,2,4-triazol-5-ylsulfanyl)furan-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-(3-fluoro-4-methoxyphenyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-({4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
2-[(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)methyl]-4,5,6,7-tetrahydro-1,3-benzothiazole
methyl 1-[(3R,5S)-1-[(4-methoxy-3-methylphenyl)methyl]-5-(4-phenylpiperazine-1-carbonyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-[(4-methylphenyl)methyl]-5-oxo-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrrolidine-3-carboxamide
4-[2-(acetamidomethyl)-1-oxa-8-azaspiro[4.5]decan-8-yl]pyrimidine-5-carboxylic acid
1-{4-[({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)methyl]piperidin-1-yl}-2-methylpropan-1-one
4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1-(propan-2-yl)pyrrolidin-2-one
6-methyl-2-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}pyridine-3-carbonitrile
N-(2-hydroxyethyl)-2-methyl-N-[(5-methylthiophen-2-yl)methyl]-1-benzofuran-7-carboxamide
3-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
7-(2-hydroxyethyl)-2-(2-methylquinolin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
6-(4-chlorophenyl)-N-cyclohexyl-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
{1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
(1S,5R)-3-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(4aS,8aR)-1-(3-hydroxypropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-N-methylpyridine-4-carboxamide
(3aR,5R,6S,7aS)-2-[(4-methanesulfonylphenyl)methyl]-octahydro-1H-isoindole-5,6-diol