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3-[(1-acetylpiperidin-4-yl)oxy]-N-[1-(2-chlorophenyl)ethyl]-4-methoxybenzamide
2-tert-butyl-N-(cyclopropylmethyl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-amine
2-[(4-methylphenyl)amino]-2-phenyl-N-{[(propan-2-yl)carbamoyl]methyl}propanamide
2-cyclopropyl-1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
2-(4-methoxy-3-methylphenyl)pyridin-3-ol
3-[1-(pyrimidin-2-yl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
1-[4-({4-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
1-(2-methylphenyl)-4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperazin-2-one
2-methoxy-1-{4-[2-(pyridin-4-ylsulfanyl)acetyl]-1,4-diazepan-1-yl}ethan-1-one
(2S,4R)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-(2,2-diphenylethyl)-N-methylpyrrolidine-2-carboxamide
{5-[4-(hydroxymethyl)phenyl]-1H-1,3-benzodiazol-2-yl}methanol
2-amino-N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}acetamide
N-(1-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-fluorobenzamide
3-{[5-(4-chloro-2-fluorophenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-ethyl-1,2,4-oxadiazole
N-ethyl-2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
N-({1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-yl}methyl)acetamide
(2S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
ethyl 4-({[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylate
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-5-methoxy-1,2-dimethyl-1H-indole-3-carboxamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
N-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
methyl 5-(cyclobutylamino)-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2-methoxyethyl)-1-{1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-{[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}-N-(propan-2-yl)piperidine-1-carboxamide
{1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidin-3-yl}methanamine
2-methoxy-1-(1'-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1-(5-propyl-1,2-oxazole-3-carbonyl)-1,2,3,6-tetrahydropyridine
N-(oxan-4-yl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-(3-hydroxy-3-phenylpropyl)-N,1-dimethyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
2-[5-(5-chloro-2-methoxyphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
ethyl 3-(2-methoxyethyl)piperidine-3-carboxylate
2-(2-hydroxyethyl)-8-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
4-(1-butyl-1H-imidazol-2-yl)-1-[4-(methylsulfanyl)benzoyl]piperidine
2-(2-fluoro-4-methylphenyl)-2-(thiomorpholin-4-yl)acetic acid
1-{1-[3-(1-methylcyclopropyl)propanoyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[2-(4-fluorophenyl)piperidin-1-yl]propan-1-one
N-(1-methyl-1H-1,2,3-triazol-4-yl)-2-[4-(quinolin-8-yl)-1H-pyrazol-1-yl]acetamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-4-(piperidin-1-yl)butanamide
4-{[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methyl}benzoic acid
5-(2-fluorophenyl)-N-[1-(pyridin-3-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[(8-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-2-methoxyacetamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(methylsulfanyl)benzamide
1-benzoyl-2-(4-fluorophenyl)piperidine
4-{[(2R,5S)-5-[(2-methylpyridin-4-yl)methyl]oxolan-2-yl]methyl}morpholine
2-[(2-ethylpyrimidin-5-yl)methyl]-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
(3S,4S)-1-{2-[(prop-2-en-1-yl)amino]benzoyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
(3aS,6aS)-2-(ethanesulfonyl)-5-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide