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ethyl 1-[2-(dimethylamino)ethyl]-5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(3S,4R)-1-[2-(2-oxopiperidin-1-yl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
1-ethyl-5-(3-oxo-1,4-diazepan-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(1S,5R)-6-methyl-3-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(furan-2-carbonyl)piperazin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
methyl 3-({5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propanoate
methyl 6-benzyl-2-[(cyclopropylmethyl)(propyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(4-ethoxy-3-methylphenyl)-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-oxobutanamide
N-[3-(4-fluorophenyl)phenyl]-1-(1,3-thiazol-2-yl)piperidine-3-carboxamide
2-[3-(dimethylamino)pyrrolidine-1-carbonyl]-6-(2,5-dimethylfuran-3-yl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-1H-indole-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-[4-(2-fluorophenyl)-1H-pyrazol-5-yl]piperidine
2-[2-methoxy-4-({3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}methyl)phenoxy]acetamide
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
5-{1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}-2-(2-methylphenyl)pyrimidine
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[4-(pyrimidin-2-yloxy)phenyl]methyl})amine
1-[2-(3-fluorophenyl)ethyl]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-6-oxopiperidine-3-carboxamide
1-benzyl-2-methyl-5-(2-methylpropanamido)-N-[3-(methylsulfanyl)propyl]-1H-1,3-benzodiazole-7-carboxamide
1-[(5-methylthiophen-2-yl)methyl]-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
5-methyl-N-[(3R,5S)-5-[(propan-2-yl)carbamoyl]-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
3-benzyl-8-[(2-hydroxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl({[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
4-(4-chlorophenoxy)-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}azepane
dimethyl({[4-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)phenyl]methyl})amine
3-(3-fluorophenyl)-4-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperazin-2-one
4-chloro-2-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1H-indole
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-6-oxo-N-(oxolan-2-ylmethyl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
5-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
N-[5-({[3-(cyclohexyloxy)-2-hydroxypropyl]carbamoyl}amino)-2-fluorophenyl]acetamide
N-cyclopropyl-4-methoxy-2-{[1-(4,4,4-trifluorobutyl)piperidin-4-yl]oxy}benzamide
9-(2-amino-6-methylpyrimidin-4-yl)-2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
8-(1-hydroxypropan-2-yl)-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1S)-2-hydroxy-1-phenylethyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
2-{1-[(2-fluorophenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
4-[2-(2,3-dihydro-1H-inden-1-yl)acetamido]-N-phenylpiperidine-1-carboxamide
[4-(2-phenoxyethyl)-1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl]methanol
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}acetamide
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-methoxypyridine-4-carboxamide
2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[4-(4-{[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}piperidin-1-yl)phenyl]-5-phenylpentanamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-hydroxy-2-methylpropanamide
3-(2-oxoimidazolidin-1-yl)-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}benzamide
5-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]-2-methylphenol
(1R,5S,6R)-N-(furan-2-ylmethyl)-3-(1H-indol-5-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-{1-[(methylcarbamoyl)methyl]piperidin-4-yl}propanamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-3-carboxylate