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1-(3-fluorophenyl)-3-{1-[1-(1H-indol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}quinoline
4-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidine
2-[({[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]-5-methoxyphenol
N-methyl-2-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
N-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}pyrimidin-2-amine
5-[(2,3-dimethoxyphenyl)methyl]-2-(4-methoxyphenyl)-6-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-methyl-8-(2-methylpropyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,4S)-2-({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2-azabicyclo[2.2.1]heptane
3-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]phenyl}-5-cyclopropyl-1,2,4-oxadiazole
{4-[2-(2-methoxy-4-methylphenoxy)ethyl]-1,4-oxazepan-6-yl}methanol
1-(2-methoxyphenyl)-5-[3-(1H-pyrazol-4-yl)propyl]-1H-1,2,4-triazole
1-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
2-(4-{[5-(2-methylpropyl)thiophen-2-yl]methyl}morpholin-2-yl)ethan-1-ol
(1S,2S)-2-{[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]amino}cyclohexan-1-ol
2-(5-acetylthiophen-3-yl)-N-(pyridin-4-ylmethyl)acetamide
(3aR,6aR)-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,2-dimethyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-methoxy-N-{[1-(3-phenylprop-2-yn-1-yl)piperidin-3-yl]methyl}benzene-1-sulfonamide
1-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]pyrrolidin-3-amine
6-(1-{furo[3,2-c]pyridin-4-yl}piperidin-3-yl)-2-phenyl-3,4-dihydropyrimidin-4-one
(2R,3R,6R)-3-(4-methylphenyl)-5-(pyridin-3-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2H-1,3-benzodioxol-4-ylmethyl)-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[2-fluoro-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
5-{1-[(2,4-dimethoxy-3-methylphenyl)methyl]piperidin-4-yl}-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
2-(adamantan-1-yl)-N-[3-(dimethylamino)-2-methylpropyl]-4-hydroxypyrimidine-5-carboxamide
3-chloro-N-cyclopentyl-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
ethyl 2-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-1,3-oxazole-4-carboxylate
1-[(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}thiophen-3-yl)methyl]piperidine
1-[(3-fluorophenyl)methyl]-N-[3-(1H-indol-1-yl)propyl]-6-oxopiperidine-3-carboxamide
2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-3-yl)-1,3-benzoxazole
4-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-1,2-dihydroquinolin-2-one
{1-[4-(azepan-1-ylmethyl)benzoyl]-3-ethylpiperidin-3-yl}methanol
5-(2,6-difluorophenoxymethyl)-N-(3-phenylpropyl)-1,2-oxazole-3-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aR,8aR)-4-[(2,6-difluoro-3-methoxyphenyl)methyl]-octahydro-2H-1,4-benzoxazine
4-(1H-imidazol-1-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]butan-1-one
N2,N4,N4,5-tetramethyl-N2-[3-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidine-2,4-diamine
1-[5-(2-chlorophenyl)furan-2-carbonyl]-3-(hydroxymethyl)piperidin-3-ol
4-[(3-fluoro-2,4-dimethylphenyl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-methyl-8-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]propan-1-one
1-tert-butyl-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]pyrrolidin-2-one
2-(2,4-dimethylphenyl)-2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
1-(4-ethylpiperazin-1-yl)-3-[3-(1,2-oxazinan-2-ylmethyl)phenoxy]propan-2-ol
2-[1-(2,2-dimethylpropyl)-4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
4'-(3-phenylpropyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-(2-methylpropyl)-3-(1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazol-2-yl)-1H-pyrazole
7-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]sulfonyl}-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
2-(2H-1,2,3-benzotriazol-2-yl)-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]acetamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2,7-dioxo-1,3-diazepane-4-carboxamide