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4-[(benzyloxy)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-1H-1,2,3-triazole
(3S,4R)-4-(3-methoxyphenyl)-1-(2-methoxypyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
1-[3-(2-methoxybenzoyl)piperidin-1-yl]-4-phenylbutane-1,4-dione
3-{4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridin-2-ol
1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4,4-difluoropiperidine
N-[(2-methoxynaphthalen-1-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
2-benzyl-8-[2-(morpholin-3-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(2R,3R)-2-methoxy-1'-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
2-(1-tert-butyl-3-methyl-1H-1,2,4-triazol-5-yl)-3,5-difluoropyridine
(1R,2S,9R)-11-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
5-(3-fluorophenoxymethyl)-3-(2-phenylazetidine-1-carbonyl)-1H-pyrazole
N-(oxolan-2-ylmethyl)-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
3-{4-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]piperazin-1-yl}pyrazine-2-carbonitrile
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
pyridin-2-yl(1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperidin-4-yl)methanol
7-[(3-methoxyphenyl)methyl]-2-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
ethyl 4-benzyl-1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidine-4-carboxylate
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-({[(3-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)-6-methylpyridin-3-ol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-3-(piperidin-3-yl)benzamide
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyridine-2-carboxamide
N-(2-chlorophenyl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)propanamide
4-(2-fluoro-5-methylphenoxy)-1-{[3-(methylsulfanyl)phenyl]methyl}piperidine-4-carboxylic acid
6-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-4-(4-methyl-1H-imidazol-5-yl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-(2,6-dichloropyridin-4-yl)-4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
9-[2-(methylamino)pyridine-4-carbonyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-N-[(4-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)-2-oxo-1,2-dihydropyridine-4-carboxamide
3-(azepane-1-carbonyl)-N-[(3-chlorophenyl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)azetidin-3-yl]-1H-1,3-benzodiazole
3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]propan-1-one
2-{2-oxo-2-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1,2-benzothiazol-3-one
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-4-ylmethyl)piperazine
N-{2-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
3-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
1-(3-chloro-2-ethoxyphenyl)-3-{2-[(2R)-pyrrolidin-2-yl]ethyl}urea
9-ethyl-4-(3-hydroxy-1,2-oxazole-5-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(4-methoxyphenyl)-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
4-[3-(dimethyl-1,2-oxazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N,N-dimethyl-5,6,7,8-tetrahydroquinazolin-2-amine
3-[1-(4-acetamido-3-methoxyphenyl)-3,5-dimethyl-1H-pyrazol-4-yl]propanoic acid
1-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
(4aR,8aR)-2-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-[3-(morpholin-4-yl)propyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}urea
2-[4-methyl-6-({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)pyrimidin-2-yl]phenol
N-({7-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-sulfonamide
methyl 5-[(adamantan-2-yl)amino]-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-({[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(benzyl)amino)ethan-1-ol