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N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
ethyl 4-{6-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
(1R)-3-methyl-1-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]butan-1-amine
{5-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]furan-2-yl}methanol
N-[2-(1H-indol-1-yl)ethyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
4-(2-cyclopropyl-1H-imidazol-1-yl)-2-(pyrrolidin-1-yl)benzamide
4-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-(4-{[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)amino]methyl}phenyl)pyrrolidin-2-one
N-(naphthalen-1-ylmethyl)-1,4-dioxane-2-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(pyridin-4-ylmethyl)acetamide
2-[5-(2-methyl-4,5,6,7-tetrahydro-2H-indazol-3-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
3-(1-butyl-1H-imidazol-2-yl)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]piperidine
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2-(morpholin-3-yl)acetamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-(5-methoxy-2-{[methyl(oxan-4-ylmethyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
4-{2-[(2-amino-6-methylpyrimidin-4-yl)amino]-1-hydroxyethyl}phenol
3-[(2,2-diethylcyclopropyl)methyl]-1-(3-methyl-1,2,4-thiadiazol-5-yl)urea
3-{2-[4-(2,4-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
3-(1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxyphenyl}-N-methylformamido)propanamide
1-(2-ethoxyethyl)-N-[(3S,5S)-5-(ethylcarbamoyl)-1-methylpyrrolidin-3-yl]-3-methyl-1H-pyrazole-5-carboxamide
6-[2-(diethylamino)-2-(furan-2-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-5-methyl-1H-pyrazole-4-carboxamide
6-ethyl-2-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrimidin-4-amine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
ethyl 1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
methyl 3-benzamido-6-{[benzyl(methyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
2-methoxy-6-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
4-chloro-5-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-5-(1H-indol-1-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
{[3-(4-methanesulfonylphenyl)phenyl]methyl}(prop-2-en-1-yl)amine
3,5-dichloro-N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-4-methylbenzamide
4-{2-[1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-2-yl]ethyl}morpholine
N,N-dimethyl-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine-1-carboxamide
(1S,5R)-6-(2,5-dimethylfuran-3-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2-dihydroquinoxalin-2-one
1-{[1-benzyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
1-cyclohexyl-6-(pyridin-2-ylmethoxy)-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1,4-diazepan-2-one
(3-chlorophenyl)[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]methanol
[3-(2-phenylethyl)-1-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-yl]methanol
(2S,4R)-4-amino-1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-N-methylpyrrolidine-2-carboxamide
ethyl 7-[(2-phenoxyethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
2-[5-methyl-2-oxo-4-(quinoline-3-carbonyl)piperazin-1-yl]benzonitrile
methyl (2S,4R)-4-({[2-(4-fluorophenyl)ethyl]carbamoyl}amino)-1-methylpyrrolidine-2-carboxylate
1-[3-(methylsulfanyl)propyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
4-({1-[2-(pyridin-3-yl)acetyl]piperidin-3-yl}methyl)benzoic acid
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][(1,5-dimethyl-1H-indazol-3-yl)methyl]amine
8-[(2-aminopyridin-3-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
4-(1,3-benzothiazol-2-yl)-2-{[(diphenylmethyl)amino]methyl}phenol