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(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(furan-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(4-fluorophenyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
2-(4-hydroxyphenyl)-1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]ethan-1-one
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-(2-fluorophenyl)-1-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-5-yl]ethan-1-one
N-[2-(1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethyl]acetamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-methyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(1H-imidazol-4-yl)-N-[(4-methylphenyl)methyl]acetamide
N-[2-(4-fluorophenyl)-2-hydroxyethyl]-4-(piperidin-1-ylmethyl)benzamide
5-(propan-2-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl})methylamine
(1S,5R)-3-methyl-6-(2,4,6-trimethylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
4-(azepan-1-yl)-N-[2-(2-methoxyphenyl)ethyl]pyridine-2-carboxamide
3-{5-[4-(1H-pyrazol-1-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]methylamine
3-chloro-5-({3-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)pyridine
(3S,5R)-5-[(6-methylpyridin-3-yl)carbamoyl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
(1S,5R)-6-(1H-indole-5-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[3-(1H-pyrazol-1-yl)propyl]amine
(1R,2S,9R)-11-[(2S)-2-methoxy-2-phenylacetyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-methyl-5-propyl-1-benzofuran-2-carboxamide
(5S)-5-[({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(pyridin-3-ylmethyl)amino)methyl]pyrrolidin-2-one
1-{2,7-diazaspiro[4.5]decan-7-yl}-4,4,4-trifluorobutan-1-one
2-(1H-1,3-benzodiazol-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}propanamide
methyl 4-[(1R,9S)-5-amino-4-cyano-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-trien-3-yl]-1H-pyrazole-3-carboxylate
2-methyl-6-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-4H-pyran-4-one
1-methyl-4-(1-{1-[4-(trifluoromethyl)benzoyl]piperidin-4-yl}ethyl)piperazine
2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoic acid
N-{2-[cyclopentyl(methyl)amino]ethyl}-N,4-dimethylquinazolin-2-amine
(2S,4R)-4-amino-1-{[5-(4-chlorophenoxy)-1,3-dimethyl-1H-pyrazol-4-yl]methyl}-N-methylpyrrolidine-2-carboxamide
2-(cyclopropylmethyl)-7-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-cyclohexyl-3-{[2-(1H-1,2,4-triazol-3-yl)phenyl]formamido}propanamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-(4-benzylpiperazin-1-yl)propan-1-one
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1-one
2-[4-(1-methoxyethyl)phenyl]-5-(piperidin-1-ylmethyl)pyridine
[(3R,4R)-1-(1-methyl-1H-pyrazole-5-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1,5-dimethyl-4-({3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-pyrazole
(2S,4R)-N-cyclopropyl-4-[(4-fluorophenyl)sulfanyl]-1-[(4-methoxynaphthalen-1-yl)methyl]pyrrolidine-2-carboxamide
6-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-methyl-8-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-ylmethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{[4-(5-methylfuran-2-yl)phenyl]methyl}-4-[2-(methylsulfanyl)ethyl]piperazine
methyl 6-{[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}pyridine-2-carboxylate
2-chloro-5-[3-(1H-pyrazol-3-yl)phenyl]benzoic acid
1-(1,4-dithiepan-6-yl)-4-[(4-fluorophenyl)methyl]piperidine
N3-[(2-chlorophenyl)methyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[(cyclopropylmethyl)sulfanyl]-1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
N-[2-(3-fluorophenyl)ethyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide