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5-(2-cyclopentylacetamido)-1-methyl-N-[2-(morpholin-4-yl)ethyl]-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
2-{3-[5-(4-methylphenyl)furan-2-yl]propanoyl}-2,7-diazaspiro[4.5]decan-6-one
[(1-cyclohexylpiperidin-3-yl)methyl][3-(methylsulfanyl)propyl](pyridin-3-ylmethyl)amine
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(3-methoxypropyl)amine
3-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]propanamide
(1S,5R)-3-(naphthalen-1-ylmethyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
6-[(2-fluorophenyl)methoxy]-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
methyl 4-({[(4-acetylmorpholin-2-yl)methyl]carbamoyl}amino)-3-chlorobenzoate
3-[(3R,4S)-1-[(5-chlorothiophen-2-yl)sulfonyl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
4-{4-[(2-aminopyrimidin-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-4-oxobutanoic acid
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-decahydro-2,7-naphthyridine-2-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]ethan-1-one
3-[(3-cyclopropyl-1H-pyrazol-5-yl)formamido]-N-(1,3-thiazol-2-yl)propanamide
(3S,4S)-1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
3-{4-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
9-(3-methoxy-2-methylbenzoyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-[(2-{4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}ethyl)sulfanyl]-1H-1,2,3-triazole
3-(2,5-dichlorophenyl)-6-methylpyridin-2-amine
1-ethyl-4-(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)piperazine
5-{6-amino-5-cyano-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]pyridin-2-yl}thiophene-3-carboxylic acid
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(propan-2-yl)-1H-1,3-benzodiazole
3-[2-(piperidin-2-yl)ethyl]-5-[5-(propan-2-yl)pyrimidin-4-yl]phenol
(1R,3R,5S)-3-(4-methoxyphenyl)-8-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-8-azabicyclo[3.2.1]octane
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
4-{4-[4-(2-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
methyl 4-{[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]methyl}benzoate
N-ethyl-1-[(2-methoxynaphthalen-1-yl)methyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-(pyrrolidin-3-yl)benzamide
3-(2-methoxyphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
4-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl]-1-(4-hydroxyphenyl)pyrrolidin-2-one
(1R,9aR)-1-[2-methyl-4-(pyrrolidin-1-ylmethyl)phenoxymethyl]-octahydro-1H-quinolizine
1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,2-dihydroquinolin-2-one
5-(hydroxymethyl)-2-methyl-4-({4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}methyl)pyridin-3-ol
2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(2-phenylethyl)acetamide
1-[(2,3-difluorophenyl)methyl]-3-{[(2,2-dimethylpropyl)amino]methyl}-3-hydroxypiperidin-2-one
(3aR,5S,6S,7aS)-2-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
N-{[2-(2,5-dimethoxyphenyl)-6-oxo-1,6-dihydropyrimidin-4-yl]methyl}acetamide
3-[1-(1-cyclobutanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-(3-fluorophenyl)urea
4-(5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzoyl)thiomorpholine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(ethylcarbamoyl)piperidine-3-carboxylate
4-benzyl-3-ethyl-1-[(4-methoxypyridin-2-yl)methyl]-1,4-diazepan-5-one
N,N-diethyl-1-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
2-{2-oxo-4-[3-(pyridin-3-yl)propanoyl]piperazin-1-yl}benzonitrile
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[3-(1H-pyrazol-1-yl)propyl]amine
7-[ethoxy(phenyl)methyl]-4-[3-(1H-pyrazol-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(carbamoylmethyl)-N-(4-ethenylphenyl)piperidine-1-carboxamide
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-(oxan-2-ylmethoxy)ethan-1-one
1-[(3-chlorophenyl)methyl]-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)-N-(2-phenylphenyl)pyrrolidine-1-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine