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1-(5-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
4-(oxolan-3-yl)-1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazole
N-[(2,6-difluorophenyl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
3-[(2-phenylquinazolin-4-yl)methyl]-1λ6-thiane-1,1-dione
N-(furan-2-ylmethyl)-1-methyl-N-(prop-2-en-1-yl)-1H-indole-2-carboxamide
7-(cyclobutylmethyl)-2-(5-methyl-1,2,4-oxadiazol-3-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(dimethylamino)ethyl]-5-(propane-2-sulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
methyl 5-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
({4-cyclopropyl-5-[1-(morpholine-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-[(1r,4r)-4-hydroxycyclohexyl]propanamide
3-(benzyloxy)-1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}azetidine
1-(2-ethoxyethyl)-N-[(6-methylpyridin-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
1-(4-{[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
5-[1-(2-fluorophenyl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]piperidin-2-one
2-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)-1,2-oxazinane
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1,4-dimethylpiperidine-4-carboxamide
1-(4-fluorophenyl)-4-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine
9-(9H-purin-6-yl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2,5-dimethyl-3-{4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}pyrazine
N-(2-{1-[4-(methylsulfanyl)benzenesulfonyl]piperidin-2-yl}ethyl)acetamide
4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-(trifluoromethyl)morpholine
N-cyclopropyl-2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}acetamide
N-methyl-N-(2-{4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-1,2,3-triazol-1-yl}ethyl)methanesulfonamide
(3aR,7aS)-2-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-({methyl[1-(2-phenylethyl)piperidin-3-yl]amino}methyl)pyridin-2-amine
4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N'-[2-(azepan-1-yl)ethyl]-N-(2-ethoxyphenyl)-N'-ethylpropanediamide
propan-2-yl (4aS,7aR)-6,6-dioxo-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
4-(cyclopropylmethyl)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3-(propan-2-yl)-1,4-diazepan-5-one
5-propyl-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1,2-oxazole-3-carboxamide
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(quinoxalin-2-ylmethyl)amine
4-(piperidin-3-yl)-N-[2-(pyridin-3-yl)ethyl]benzamide
1-[3-(4-fluorophenyl)phenyl]-N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-amine
N'1-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}cyclopropane-1,1-dicarboxamide
2-amino-6-(3-hydroxyphenyl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
N-methyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(quinolin-6-ylmethyl)piperidine-3-carboxamide
6-(2,5-dimethylfuran-3-yl)-2-(3-hydroxyazetidine-1-carbonyl)-7-(3-methylbut-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-(6-phenoxypyridin-3-yl)-1-[2-(1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxamide
3,4-dimethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)benzamide
(3aR,6aR)-2-[2-(2,3-dimethylphenoxy)acetyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 2-{8-[(3-hydroxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
8-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-(4-ethyl-5-methylpyrimidin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(ethylamino)-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-methyl-1,3-thiazole-5-carboxamide
N,1,6-trimethyl-N-[(1-methylpiperidin-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-({1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl}methyl)benzamide
N,N-dimethyl-1-({1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazol-5-yl}methyl)pyrrolidin-3-amine
4-[5-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one